Long-term efficacy and safety of iloperidone: an update.

Article Details

Citation

Rado JT, Janicak PG

Long-term efficacy and safety of iloperidone: an update.

Neuropsychiatr Dis Treat. 2014 Feb 26;10:409-15. doi: 10.2147/NDT.S37824. eCollection 2014.

PubMed ID
24600226 [ View in PubMed
]
Abstract

Schizophrenia is a devastating neuropsychiatric disease with a worldwide prevalence of approximately 0.5%-1%. Since many patients do not achieve adequate symptom relief from available agents, alternate pharmacotherapeutic approaches are needed. In this context, iloperidone was recently approved by the US Food and Drug Administration for the treatment of schizophrenia. This paper first reviews its pharmacodynamic and pharmacokinetic profiles, emphasizing their clinical relevance. Next, it summarizes the literature on its acute and maintenance efficacy, safety, and tolerability. It then considers pharmacogenetic data which may help to predict response and risk of cardiac arrhythmias with this agent. Finally, it critically positions iloperidone relative to other first- and second-generation antipsychotics.

DrugBank Data that Cites this Article

Drugs
Drug Targets
DrugTargetKindOrganismPharmacological ActionActions
Iloperidone5-hydroxytryptamine receptor 1AProteinHumans
Unknown
Antagonist
Details
Iloperidone5-hydroxytryptamine receptor 2AProteinHumans
Yes
Antagonist
Details
Iloperidone5-hydroxytryptamine receptor 2CProteinHumans
Unknown
Antagonist
Details
Iloperidone5-hydroxytryptamine receptor 6ProteinHumans
Unknown
Antagonist
Details
IloperidoneAlpha-1A adrenergic receptorProteinHumans
Unknown
Antagonist
Details
IloperidoneAlpha-2A adrenergic receptorProteinHumans
Unknown
Antagonist
Details
IloperidoneAlpha-2B adrenergic receptorProteinHumans
Unknown
Antagonist
Details
IloperidoneAlpha-2C adrenergic receptorProteinHumans
Unknown
Antagonist
Details
IloperidoneBeta-1 adrenergic receptorProteinHumans
Unknown
Antagonist
Details
IloperidoneBeta-2 adrenergic receptorProteinHumans
Unknown
Antagonist
Details
IloperidoneD(1A) dopamine receptorProteinHumans
Unknown
Antagonist
Details
IloperidoneD(1B) dopamine receptorProteinHumans
Unknown
Antagonist
Details
IloperidoneD(2) dopamine receptorProteinHumans
Yes
Antagonist
Details
IloperidoneD(3) dopamine receptorProteinHumans
Unknown
Antagonist
Details
IloperidoneD(4) dopamine receptorProteinHumans
Unknown
Antagonist
Details
IloperidoneHistamine H1 receptorProteinHumans
Unknown
Antagonist
Details