Angiotensin 2 Receptor Blocker

Name
Angiotensin 2 Receptor Blocker
Accession Number
DBCAT003287
Description

Not Available

Drugs
DrugDrug Description
ValsartanAn angiotensin-receptor blocker used to manage hypertension alone or in combination with other antihypertensive agents and to manage heart failure in patients who are intolerant to ACE inhibitors.
OlmesartanAn angiotensin receptor blocker (ARB) used in the treatment of hypertension.
LosartanAn angiotensin receptor blocker used to treat hypertension and diabetic nephropathy, and is used to reduce the risk of stroke.
EprosartanAn ARB used to treat hypertension, diabetic nephropathy, and congestive heart failure.
TelmisartanAn ARB used to treat hypertension, diabetic nephropathy, and congestive heart failure.
IrbesartanAn angiotensin receptor blocker used to treat hypertension, delay progression of diabetic nephropathy, and treat congestive heart failure.
Azilsartan medoxomilAn angiotensin II receptor blocker used to treat hypertension alone or in combination with other antihypertensive agents, such as chlorthalidone.
CandesartanAn angiotensin-receptor blocker indicated in the treatment of hypertension.
Candesartan cilexetilAn angiotensin receptor blocker used to treat hypertension, systolic hypertension, left ventricular hypertrophy, and delay progression of diabetic nephropathy.
SparsentanAn endothelin and angiotensin II receptor antagonist indicated to reduce proteinuria in adults with primary immunoglobulin A nephropathy at risk of rapid disease progression.
Drugs & Drug Targets
DrugTargetType
ValsartanType-1 angiotensin II receptortarget
ValsartanCytochrome P450 2C9enzyme
ValsartanSolute carrier organic anion transporter family member 1B3transporter
ValsartanSolute carrier organic anion transporter family member 1B1transporter
ValsartanATP-binding cassette sub-family C member 2transporter
OlmesartanType-1 angiotensin II receptortarget
OlmesartanATP-binding cassette sub-family C member 2transporter
OlmesartanSolute carrier organic anion transporter family member 1B3transporter
OlmesartanSolute carrier organic anion transporter family member 1B1transporter
OlmesartanBile salt export pumptransporter
LosartanType-1 angiotensin II receptortarget
LosartanCytochrome P450 3A4enzyme
LosartanCytochrome P450 2C9enzyme
LosartanATP-dependent translocase ABCB1transporter
LosartanSolute carrier family 22 member 6transporter
LosartanUDP-glucuronosyltransferase 1A1enzyme
LosartanUDP-glucuronosyltransferase 1A3enzyme
LosartanUDP-glucuronosyltransferase 1A10enzyme
LosartanUDP-glucuronosyltransferase 2B7enzyme
LosartanUDP-glucuronosyltransferase 2B17enzyme
LosartanCytochrome P450 2C19enzyme
LosartanAlbumincarrier
LosartanSolute carrier family 22 member 12transporter
LosartanSolute carrier family 2, facilitated glucose transporter member 9transporter
LosartanBile salt export pumptransporter
LosartanCytochrome P450 2C8enzyme
LosartanErythropoietin receptortarget
EprosartanType-1 angiotensin II receptortarget
EprosartanATP-binding cassette sub-family C member 2transporter
TelmisartanType-1 angiotensin II receptortarget
TelmisartanPeroxisome proliferator-activated receptor gammatarget
TelmisartanATP-dependent translocase ABCB1transporter
TelmisartanATP-binding cassette sub-family C member 2transporter
TelmisartanBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TelmisartanCytochrome P450 2C19enzyme
TelmisartanBile salt export pumptransporter
TelmisartanUDP-glucuronosyltransferase 1A3enzyme
IrbesartanType-1 angiotensin II receptortarget
IrbesartanTranscription factor Juntarget
IrbesartanCytochrome P450 2C9enzyme
IrbesartanCytochrome P450 2C8enzyme
IrbesartanUDP-glucuronosyltransferase 1A3enzyme
IrbesartanProstaglandin G/H synthase 1enzyme
IrbesartanCytochrome P450 3A4enzyme
IrbesartanAlbumincarrier
Irbesartanalpha1-acid glycoproteincarrier
Azilsartan medoxomilType-1 angiotensin II receptortarget
Azilsartan medoxomilAlbumincarrier
Azilsartan medoxomilCytochrome P450 2C9enzyme
Azilsartan medoxomilCytochrome P450 2C8enzyme
Azilsartan medoxomilCytochrome P450 2B6enzyme
Azilsartan medoxomilATP-dependent translocase ABCB1transporter
CandesartanType-1 angiotensin II receptortarget
CandesartanCytochrome P450 2C8enzyme
CandesartanCytochrome P450 2C9enzyme
CandesartanATP-dependent translocase ABCB1transporter
CandesartanUDP-glucuronosyltransferase 1A3enzyme
CandesartanProstaglandin G/H synthase 1enzyme
CandesartanSolute carrier organic anion transporter family member 1B1transporter
Candesartan cilexetilType-1 angiotensin II receptortarget
Candesartan cilexetilCytochrome P450 2C8enzyme
Candesartan cilexetilCytochrome P450 2C9enzyme
Candesartan cilexetilATP-dependent translocase ABCB1transporter
Candesartan cilexetilUDP-glucuronosyltransferase 1A3enzyme
Candesartan cilexetilProstaglandin G/H synthase 1enzyme
SparsentanEndothelin-1 receptortarget
SparsentanType-2 angiotensin II receptortarget
SparsentanCytochrome P450 3A4enzyme
SparsentanCytochrome P450 2B6enzyme
SparsentanCytochrome P450 2C9enzyme
SparsentanCytochrome P450 2C19enzyme
SparsentanATP-dependent translocase ABCB1transporter
SparsentanBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
SparsentanSolute carrier organic anion transporter family member 1B3transporter
SparsentanOrganic anion transporter 3transporter
SparsentanType-1 angiotensin II receptortarget