Antipsychotic Medications

Article Details

Citation

Chokhawala K, Stevens L

Antipsychotic Medications

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PubMed ID
30137788 [ View in PubMed
]
Abstract

First-generation antipsychotics are dopamine receptor antagonists (DRA) and are known as typical antipsychotics. They include phenothiazines (trifluoperazine, perphenazine, prochlorperazine, acetophenazine, triflupromazine, mesoridazine), butyrophenones (haloperidol), thioxanthenes (thiothixene, chlorprothixene), dibenzoxazepines (loxapine), dihydroindoles (molindone), and diphenylbutylpiperidines (pimozide).[1][2][3]

DrugBank Data that Cites this Article

Drug Targets
DrugTargetKindOrganismPharmacological ActionActions
TriflupromazineDopamine D1 receptorProteinHumans
Yes
Antagonist
Details
TriflupromazineDopamine D2 receptorProteinHumans
Yes
Antagonist
Details