Angiotensin II AT1 receptor antagonists. Clinical implications of active metabolites.

Article Details

Citation

Schmidt B, Schieffer B

Angiotensin II AT1 receptor antagonists. Clinical implications of active metabolites.

J Med Chem. 2003 Jun 5;46(12):2261-70.

PubMed ID
12773029 [ View in PubMed
]
Abstract

Not Available

DrugBank Data that Cites this Article

Binding Properties
DrugTargetPropertyMeasurementpHTemperature (°C)
TasosartanType-1 angiotensin II receptorIC 50 (nM)32N/AN/ADetails
ValsartanType-1 angiotensin II receptorKi (nM)4700N/AN/ADetails