Neuronal nicotinic acetylcholine receptors as targets for drug discovery.

Article Details

Citation

Holladay MW, Dart MJ, Lynch JK

Neuronal nicotinic acetylcholine receptors as targets for drug discovery.

J Med Chem. 1997 Dec 19;40(26):4169-94.

PubMed ID
9435889 [ View in PubMed
]
Abstract

Not Available

DrugBank Data that Cites this Article

Binding Properties
DrugTargetPropertyMeasurementpHTemperature (°C)
NicotineNeuronal acetylcholine receptor subunit beta-2EC 50 (nM)4000N/AN/ADetails
RivaniclineNeuronal acetylcholine receptor subunit beta-2EC 50 (nM)4300N/AN/ADetails