Neuronal nicotinic acetylcholine receptors: structural revelations, target identifications, and therapeutic inspirations.
Article Details
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Jensen AA, Frolund B, Liljefors T, Krogsgaard-Larsen P
Neuronal nicotinic acetylcholine receptors: structural revelations, target identifications, and therapeutic inspirations.
J Med Chem. 2005 Jul 28;48(15):4705-45.
- PubMed ID
- 16033252 [ View in PubMed]
- Abstract
Not Available
DrugBank Data that Cites this Article
- Binding Properties
Drug Target Property Measurement pH Temperature (°C) Mecamylamine Neuronal acetylcholine receptor subunit alpha-2 IC 50 (nM) 16000 N/A N/A Details Mecamylamine Neuronal acetylcholine receptor subunit alpha-2 IC 50 (nM) 3100 N/A N/A Details Mecamylamine Neuronal acetylcholine receptor subunit beta-2 IC 50 (nM) 280 N/A N/A Details Nicotine Neuronal acetylcholine receptor subunit beta-2 EC 50 (nM) 132000 N/A N/A Details