Neuronal nicotinic acetylcholine receptors: structural revelations, target identifications, and therapeutic inspirations.

Article Details

Citation

Jensen AA, Frolund B, Liljefors T, Krogsgaard-Larsen P

Neuronal nicotinic acetylcholine receptors: structural revelations, target identifications, and therapeutic inspirations.

J Med Chem. 2005 Jul 28;48(15):4705-45.

PubMed ID
16033252 [ View in PubMed
]
Abstract

Not Available

DrugBank Data that Cites this Article

Binding Properties
DrugTargetPropertyMeasurementpHTemperature (°C)
MecamylamineNeuronal acetylcholine receptor subunit alpha-2IC 50 (nM)16000N/AN/ADetails
MecamylamineNeuronal acetylcholine receptor subunit alpha-2IC 50 (nM)3100N/AN/ADetails
MecamylamineNeuronal acetylcholine receptor subunit beta-2IC 50 (nM)280N/AN/ADetails
NicotineNeuronal acetylcholine receptor subunit beta-2EC 50 (nM)132000N/AN/ADetails