Probing the molecular basis of resistance to pyrimethamine by site-directed mutagenesis.
Article Details
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Wagner CR, Benkovic SJ
Probing the molecular basis of resistance to pyrimethamine by site-directed mutagenesis.
J Med Chem. 1992 Jul 24;35(15):2912-5.
- PubMed ID
- 1495020 [ View in PubMed]
- Abstract
Not Available
DrugBank Data that Cites this Article
- Binding Properties
Drug Target Property Measurement pH Temperature (°C) Pyrimethamine Dihydrofolate reductase Kd (nM) 13 N/A N/A Details Pyrimethamine Dihydrofolate reductase Ki (nM) 10 N/A N/A Details Pyrimethamine Dihydrofolate reductase Ki (nM) 20 N/A N/A Details Pyrimethamine Dihydrofolate reductase Kd (nM) 16 N/A N/A Details Pyrimethamine Dihydrofolate reductase Ki (nM) 2 N/A N/A Details Pyrimethamine Dihydrofolate reductase Ki (nM) 5.2 N/A N/A Details Pyrimethamine Dihydrofolate reductase Kd (nM) 1.4 N/A N/A Details Pyrimethamine Dihydrofolate reductase Ki (nM) 1.2 N/A N/A Details Pyrimethamine Dihydrofolate reductase Ki (nM) 0.19 N/A N/A Details Pyrimethamine Dihydrofolate reductase Kd (nM) 1.5 N/A N/A Details