Molecular biology of 5-HT receptors.

Article Details

Citation

Boess FG, Martin IL

Molecular biology of 5-HT receptors.

Neuropharmacology. 1994 Mar-Apr;33(3-4):275-317.

PubMed ID
7984267 [ View in PubMed
]
Abstract

Not Available

DrugBank Data that Cites this Article

Binding Properties
DrugTargetPropertyMeasurementpHTemperature (°C)
Buspirone5-hydroxytryptamine receptor 1AKi (nM)3.98N/AN/ADetails
Buspirone5-hydroxytryptamine receptor 1AKi (nM)77.62N/AN/ADetails
Buspirone5-hydroxytryptamine receptor 1AKi (nM)19.05N/AN/ADetails
Buspirone5-hydroxytryptamine receptor 1AKi (nM)21.37N/AN/ADetails
Buspirone5-hydroxytryptamine receptor 1AKi (nM)15.13N/AN/ADetails
Buspirone5-hydroxytryptamine receptor 1AKi (nM)213.79N/AN/ADetails
Cyproheptadine5-hydroxytryptamine receptor 2AKi (nM)2.88N/AN/ADetails
Ergotamine5-hydroxytryptamine receptor 1FKi (nM)169.82N/AN/ADetails
Lysergic acid diethylamide5-hydroxytryptamine receptor 1AKi (nM)1.09N/AN/ADetails
Methysergide5-hydroxytryptamine receptor 1AKi (nM)16.98N/AN/ADetails
Methysergide5-hydroxytryptamine receptor 1BKi (nM)25.11N/AN/ADetails
Methysergide5-hydroxytryptamine receptor 1BKi (nM)162.18N/AN/ADetails
Methysergide5-hydroxytryptamine receptor 1BKi (nM)7.58N/AN/ADetails
Methysergide5-hydroxytryptamine receptor 1EKi (nM)229.08N/AN/ADetails
Methysergide5-hydroxytryptamine receptor 1EKi (nM)323.59N/AN/ADetails
Methysergide5-hydroxytryptamine receptor 1EKi (nM)218.77N/AN/ADetails
Methysergide5-hydroxytryptamine receptor 1FKi (nM)33.88N/AN/ADetails
Methysergide5-hydroxytryptamine receptor 2AKi (nM)3.31N/AN/ADetails
Mianserin5-hydroxytryptamine receptor 1AKi (nM)512.86N/AN/ADetails
Mianserin5-hydroxytryptamine receptor 1AKi (nM)398.1N/AN/ADetails
Mianserin5-hydroxytryptamine receptor 1FKi (nM)12.58N/AN/ADetails
Pindolol5-hydroxytryptamine receptor 1AKi (nM)17.78N/AN/ADetails
Pindolol5-hydroxytryptamine receptor 1AKi (nM)37.15N/AN/ADetails
Pindolol5-hydroxytryptamine receptor 1AKi (nM)33.11N/AN/ADetails
Pindolol5-hydroxytryptamine receptor 1AKi (nM)28.18N/AN/ADetails
Pindolol5-hydroxytryptamine receptor 1AKi (nM)61.65N/AN/ADetails
Propranolol5-hydroxytryptamine receptor 1BKi (nM)2691.53N/AN/ADetails
Propranolol5-hydroxytryptamine receptor 1BKi (nM)>10000N/AN/ADetails
Propranolol5-hydroxytryptamine receptor 1BKi (nM)630.95N/AN/ADetails
Propranolol5-hydroxytryptamine receptor 1BKi (nM)56.23N/AN/ADetails
Sumatriptan5-hydroxytryptamine receptor 1AKi (nM)1023.29N/AN/ADetails
Sumatriptan5-hydroxytryptamine receptor 1AKi (nM)257.03N/AN/ADetails
Sumatriptan5-hydroxytryptamine receptor 1BKi (nM)7.76N/AN/ADetails
Sumatriptan5-hydroxytryptamine receptor 1BKi (nM)9.33N/AN/ADetails
Sumatriptan5-hydroxytryptamine receptor 1BKi (nM)10.96N/AN/ADetails
Sumatriptan5-hydroxytryptamine receptor 1BKi (nM)1.99N/AN/ADetails
Sumatriptan5-hydroxytryptamine receptor 1BKi (nM)61.65N/AN/ADetails
Sumatriptan5-hydroxytryptamine receptor 1DKi (nM)3.71N/AN/ADetails
Sumatriptan5-hydroxytryptamine receptor 1DKi (nM)3.38N/AN/ADetails
Sumatriptan5-hydroxytryptamine receptor 1FKi (nM)22.9N/AN/ADetails
Yohimbine5-hydroxytryptamine receptor 1BKi (nM)39.81N/AN/ADetails
Yohimbine5-hydroxytryptamine receptor 1BKi (nM)46.77N/AN/ADetails
Yohimbine5-hydroxytryptamine receptor 1BKi (nM)251.18N/AN/ADetails
Yohimbine5-hydroxytryptamine receptor 1BKi (nM)26.91N/AN/ADetails
Yohimbine5-hydroxytryptamine receptor 1BKi (nM)40.73N/AN/ADetails
Yohimbine5-hydroxytryptamine receptor 1BKi (nM)5.01N/AN/ADetails
Yohimbine5-hydroxytryptamine receptor 1DKi (nM)15.84N/AN/ADetails
Yohimbine5-hydroxytryptamine receptor 1DKi (nM)58.88N/AN/ADetails
Yohimbine5-hydroxytryptamine receptor 1DKi (nM)47.86N/AN/ADetails
Yohimbine5-hydroxytryptamine receptor 1DKi (nM)21.87N/AN/ADetails