The many roles for fluorine in medicinal chemistry.
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Hagmann WK
The many roles for fluorine in medicinal chemistry.
J Med Chem. 2008 Aug 14;51(15):4359-69. doi: 10.1021/jm800219f. Epub 2008 Jun 21.
- PubMed ID
- 18570365 [ View in PubMed]
- Abstract
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- Binding Properties
Drug Target Property Measurement pH Temperature (°C) Aprepitant Neurokinin 1 receptor IC 50 (nM) 0.09 N/A N/A Details Sitagliptin Dipeptidyl peptidase 4 IC 50 (nM) 18 N/A N/A Details