Atropisomeric derivatives of 2',6'-disubstituted (R)-11-phenylaporphine: selective serotonin 5-HT(7) receptor antagonists.

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Linnanen T, Brisander M, Unelius L, Rosqvist S, Nordvall G, Hacksell U, Johansson AM

Atropisomeric derivatives of 2',6'-disubstituted (R)-11-phenylaporphine: selective serotonin 5-HT(7) receptor antagonists.

J Med Chem. 2001 Apr 26;44(9):1337-40.

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11311055 [ View in PubMed

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DrugBank Data that Cites this Article

Binding Properties

Drug	Target	Property	Measurement	pH	Temperature (°C)
Apomorphine	5-hydroxytryptamine receptor 1A	Ki (nM)	296	N/A	N/A	Details
Apomorphine	Dopamine D2 receptor	Ki (nM)	41.9	N/A	N/A	Details