Identification of retinoic acid receptor beta subtype specific agonists.

Article Details

Citation

Johnson AT, Klein ES, Wang L, Pino ME, Chandraratna RA

Identification of retinoic acid receptor beta subtype specific agonists.

J Med Chem. 1996 Dec 20;39(26):5027-30.

PubMed ID
8978832 [ View in PubMed
]
Abstract

Not Available

DrugBank Data that Cites this Article

Binding Properties
DrugTargetPropertyMeasurementpHTemperature (°C)
TretinoinRetinoic acid receptor alphaKd (nM)15N/AN/ADetails
TretinoinRetinoic acid receptor alphaEC 50 (nM)459N/AN/ADetails
TretinoinRetinoic acid receptor betaKd (nM)13N/AN/ADetails
TretinoinRetinoic acid receptor betaEC 50 (nM)87N/AN/ADetails
TretinoinRetinoic acid receptor gammaKd (nM)18N/AN/ADetails
TretinoinRetinoic acid receptor gammaEC 50 (nM)20N/AN/ADetails