Carnitine palmitoyltransferase (CPT) modulators: a medicinal chemistry perspective on 35 years of research.
Article Details
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Ceccarelli SM, Chomienne O, Gubler M, Arduini A
Carnitine palmitoyltransferase (CPT) modulators: a medicinal chemistry perspective on 35 years of research.
J Med Chem. 2011 May 12;54(9):3109-52. doi: 10.1021/jm100809g. Epub 2011 Apr 19.
- PubMed ID
- 21504156 [ View in PubMed]
- Abstract
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DrugBank Data that Cites this Article
- Binding Properties
Drug Target Property Measurement pH Temperature (°C) Perhexiline Carnitine O-palmitoyltransferase 1, liver isoform IC 50 (nM) >100000 N/A N/A Details Perhexiline Carnitine O-palmitoyltransferase 2, mitochondrial IC 50 (nM) 72800 N/A N/A Details