Carnitine palmitoyltransferase (CPT) modulators: a medicinal chemistry perspective on 35 years of research.

Article Details

Citation

Ceccarelli SM, Chomienne O, Gubler M, Arduini A

Carnitine palmitoyltransferase (CPT) modulators: a medicinal chemistry perspective on 35 years of research.

J Med Chem. 2011 May 12;54(9):3109-52. doi: 10.1021/jm100809g. Epub 2011 Apr 19.

PubMed ID
21504156 [ View in PubMed
]
Abstract

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DrugBank Data that Cites this Article

Binding Properties
DrugTargetPropertyMeasurementpHTemperature (°C)
PerhexilineCarnitine O-palmitoyltransferase 1, liver isoformIC 50 (nM)>100000N/AN/ADetails
PerhexilineCarnitine O-palmitoyltransferase 2, mitochondrialIC 50 (nM)72800N/AN/ADetails