Small molecule JNK (c-Jun N-terminal kinase) inhibitors.

Article Details

Citation

Siddiqui MA, Reddy PA

Small molecule JNK (c-Jun N-terminal kinase) inhibitors.

J Med Chem. 2010 Apr 22;53(8):3005-12. doi: 10.1021/jm9003279.

PubMed ID
20146479 [ View in PubMed
]
Abstract

Not Available

DrugBank Data that Cites this Article

Binding Properties
DrugTargetPropertyMeasurementpHTemperature (°C)
PyrazolanthroneMitogen-activated protein kinase 10IC 50 (nM)90N/AN/ADetails
PyrazolanthroneMitogen-activated protein kinase 8IC 50 (nM)40N/AN/ADetails