On-chip fragment-based approach for discovery of high-affinity bivalent inhibitors.
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Miyazaki I, Simizu S, Ishida K, Osada H
On-chip fragment-based approach for discovery of high-affinity bivalent inhibitors.
Chembiochem. 2009 Mar 23;10(5):838-43. doi: 10.1002/cbic.200800704.
- PubMed ID
- 19226504 [ View in PubMed]
- Abstract
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DrugBank Data that Cites this Article
- Binding Properties
Drug Target Property Measurement pH Temperature (°C) 4-Flourobenzenesulfonamide Carbonic anhydrase 2 IC 50 (nM) 203 8.4 N/A Details 4-Flourobenzenesulfonamide Carbonic anhydrase 2 Kd (nM) 435 8.4 N/A Details