On-chip fragment-based approach for discovery of high-affinity bivalent inhibitors.

Article Details

Citation

Miyazaki I, Simizu S, Ishida K, Osada H

On-chip fragment-based approach for discovery of high-affinity bivalent inhibitors.

Chembiochem. 2009 Mar 23;10(5):838-43. doi: 10.1002/cbic.200800704.

PubMed ID
19226504 [ View in PubMed
]
Abstract

Not Available

DrugBank Data that Cites this Article

Binding Properties
DrugTargetPropertyMeasurementpHTemperature (°C)
4-FlourobenzenesulfonamideCarbonic anhydrase 2IC 50 (nM)2038.4N/ADetails
4-FlourobenzenesulfonamideCarbonic anhydrase 2Kd (nM)4358.4N/ADetails