Evolution of poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors. From concept to clinic.
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Ferraris DV
Evolution of poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors. From concept to clinic.
J Med Chem. 2010 Jun 24;53(12):4561-84. doi: 10.1021/jm100012m.
- PubMed ID
- 20364863 [ View in PubMed]
- Abstract
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DrugBank Data that Cites this Article
- Binding Properties
Drug Target Property Measurement pH Temperature (°C) Nicotinamide Poly [ADP-ribose] polymerase 1 IC 50 (nM) 210000 N/A N/A Details