Evolution of poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors. From concept to clinic.

Article Details

Citation

Ferraris DV

Evolution of poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors. From concept to clinic.

J Med Chem. 2010 Jun 24;53(12):4561-84. doi: 10.1021/jm100012m.

PubMed ID
20364863 [ View in PubMed
]
Abstract

Not Available

DrugBank Data that Cites this Article

Binding Properties
DrugTargetPropertyMeasurementpHTemperature (°C)
NicotinamidePoly [ADP-ribose] polymerase 1IC 50 (nM)210000N/AN/ADetails