Discovery of a potent, orally active, nonsteroidal androgen receptor agonist: 4-ethyl-1,2,3,4-tetrahydro-6- (trifluoromethyl)-8-pyridono[5,6-g]- quinoline (LG121071).

Article Details

Citation

Copy to clipboard

Hamann LG, Mani NS, Davis RL, Wang XN, Marschke KB, Jones TK

Discovery of a potent, orally active, nonsteroidal androgen receptor agonist: 4-ethyl-1,2,3,4-tetrahydro-6- (trifluoromethyl)-8-pyridono[5,6-g]- quinoline (LG121071).

J Med Chem. 1999 Jan 28;42(2):210-2.

PubMed ID

9925725 [ View in PubMed

]

Abstract

Not Available

DrugBank Data that Cites this Article

Binding Properties

Drug	Target	Property	Measurement	pH	Temperature (°C)
Stanolone	Androgen receptor	Ki (nM)	3	N/A	N/A	Details
Stanolone	Androgen receptor	IC 50 (nM)	0	N/A	N/A	Details
Stanolone	Androgen receptor	EC 50 (nM)	5	N/A	N/A	Details