Selective p38alpha inhibitors clinically evaluated for the treatment of chronic inflammatory disorders.

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Goldstein DM, Kuglstatter A, Lou Y, Soth MJ

Selective p38alpha inhibitors clinically evaluated for the treatment of chronic inflammatory disorders.

J Med Chem. 2010 Mar 25;53(6):2345-53. doi: 10.1021/jm9012906.

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19950901 [ View in PubMed

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DrugBank Data that Cites this Article

Binding Properties

Drug	Target	Property	Measurement	pH	Temperature (°C)
Neflamapimod	Mitogen-activated protein kinase 14	IC 50 (nM)	10	N/A	N/A	Details
PH-797804	Mitogen-activated protein kinase 14	Ki (nM)	5.8	N/A	N/A	Details