Stoichiometry of the human glycine receptor revealed by direct subunit counting.

Article Details

Citation

Durisic N, Godin AG, Wever CM, Heyes CD, Lakadamyali M, Dent JA

Stoichiometry of the human glycine receptor revealed by direct subunit counting.

J Neurosci. 2012 Sep 12;32(37):12915-20. doi: 10.1523/JNEUROSCI.2050-12.2012.

PubMed ID
22973015 [ View in PubMed
]
Abstract

The subunit stoichiometry of heteromeric glycine-gated channels determines fundamental properties of these key inhibitory neurotransmitter receptors; however, the ratio of alpha1- to beta-subunits per receptor remains controversial. We used single-molecule imaging and stepwise photobleaching in Xenopus oocytes to directly determine the subunit stoichiometry of a glycine receptor to be 3alpha1:2beta. This approach allowed us to determine the receptor stoichiometry in mixed populations consisting of both heteromeric and homomeric channels, additionally revealing the quantitative proportions for the two populations.

DrugBank Data that Cites this Article

Polypeptides
NameUniProt ID
Glycine receptor subunit betaP48167Details
Glycine receptor subunit alpha-1P23415Details