Sodium-glucose Cotransporter 2 (SGLT2) Inhibitors

Name
Sodium-glucose Cotransporter 2 (SGLT2) Inhibitors
Accession Number
DBCAT003772  (DBCAT002659, DBCAT003469, DBCAT004600)
Description

Not Available

ATC Classification
Drugs
DrugDrug Description
DapagliflozinA sodium-glucose cotransporter 2 inhibitor used in the management of type 2 diabetes mellitus.
CanagliflozinA sodium-glucose co-transporter 2 (SGLT2) inhibitor used to manage hyperglycemia in type 2 diabetes mellitus (DM). Also used to reduce the risk of major cardiovascular events in patients with established cardiovascular disease and type 2 DM.
ErtugliflozinAn SGLT2 inhibitor used to treat type 2 diabetes mellitus alone or in combination with other antidiabetic drugs.
IpragliflozinIpragliflozin is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.
SotagliflozinAn orally administered dual SGLT1/2 inhibitor used alongside insulin to improve glycemic control in patients with type 1 diabetes mellitus.
EmpagliflozinAn SGLT2 inhibitor used to manage type 2 diabetes mellitus.
LuseogliflozinAn SGLT2 inhibitor used to manage type 2 diabetes mellitus.
BexagliflozinA sodium-glucose co-transporter 2 inhibitor used to improve glycemic control in patients with type 2 diabetes mellitus.
Drugs & Drug Targets
DrugTargetType
DapagliflozinSodium/glucose cotransporter 2target
DapagliflozinCytochrome P450 1A1enzyme
DapagliflozinCytochrome P450 1A2enzyme
DapagliflozinCytochrome P450 2A6enzyme
DapagliflozinCytochrome P450 2C9enzyme
DapagliflozinCytochrome P450 2D6enzyme
DapagliflozinCytochrome P450 3A4enzyme
DapagliflozinUDP-glucuronosyltransferase 1-9enzyme
DapagliflozinUDP-glucuronosyltransferase 2B4enzyme
DapagliflozinUDP-glucuronosyltransferase 2B7enzyme
DapagliflozinP-glycoprotein 1transporter
CanagliflozinUDP-glucuronosyltransferase 1-9enzyme
CanagliflozinUDP-glucuronosyltransferase 2B4enzyme
CanagliflozinCytochrome P450 3A4enzyme
CanagliflozinSodium/glucose cotransporter 2target
CanagliflozinP-glycoprotein 1transporter
CanagliflozinCanalicular multispecific organic anion transporter 1transporter
CanagliflozinAlpha-1-acid glycoprotein 1carrier
CanagliflozinATP-binding cassette sub-family G member 2transporter
ErtugliflozinUDP-glucuronosyltransferase 1-9enzyme
ErtugliflozinUDP-glucuronosyltransferase 2B7enzyme
ErtugliflozinSodium/glucose cotransporter 2target
ErtugliflozinP-glycoprotein 1transporter
ErtugliflozinATP-binding cassette sub-family G member 2transporter
ErtugliflozinSerum albumincarrier
ErtugliflozinUDP-glucuronosyltransferase 1-1enzyme
ErtugliflozinUDP-glucuronosyltransferase 1-4enzyme
SotagliflozinUDP-glucuronosyltransferase 1-9enzyme
SotagliflozinUDP-glucuronosyltransferase 1-1enzyme
SotagliflozinUDP-glucuronosyltransferase 2B7enzyme
SotagliflozinCytochrome P450 3A4enzyme
SotagliflozinSodium/glucose cotransporter 2target
SotagliflozinSodium/glucose cotransporter 1target
SotagliflozinCytochrome P450 2D6enzyme
SotagliflozinP-glycoprotein 1transporter
SotagliflozinATP-binding cassette sub-family G member 2transporter
SotagliflozinSolute carrier organic anion transporter family member 1B1transporter
SotagliflozinSolute carrier organic anion transporter family member 1B3transporter
SotagliflozinCanalicular multispecific organic anion transporter 1transporter
EmpagliflozinSodium/glucose cotransporter 2target
EmpagliflozinUDP-glucuronosyltransferase 2B7enzyme
EmpagliflozinUDP-glucuronosyltransferase 1-3enzyme
EmpagliflozinUDP-glucuronosyltransferase 1-8enzyme
EmpagliflozinUDP-glucuronosyltransferase 1-9enzyme
EmpagliflozinP-glycoprotein 1transporter
EmpagliflozinATP-binding cassette sub-family G member 2transporter
EmpagliflozinSolute carrier family 22 member 8transporter
EmpagliflozinSolute carrier organic anion transporter family member 1B1transporter
EmpagliflozinSolute carrier organic anion transporter family member 1B3transporter
BexagliflozinUDP-glucuronosyltransferase 1-9enzyme
BexagliflozinCytochrome P450 3A4enzyme
BexagliflozinCytochrome P450 2C8enzyme
BexagliflozinCytochrome P450 2D6enzyme
BexagliflozinUDP-glucuronosyltransferase 1-1enzyme
BexagliflozinSodium/glucose cotransporter 2target
BexagliflozinP-glycoprotein 1transporter