Antidepressive Agents

Also known as: Antidepressant / Antidepressants / Antidepressive Agent / Antidepressant (substance) / Medicinal product acting as antidepressant agent (product)

DrugDrug NameDrug Description
DB09128BrexpiprazoleA serotonin–dopamine activity modulator used in the treatment of major depressive disorder as an adjunct, schizophrenia, and agitation associated with dementia due to Alzheimer’s disease.
DB01267PaliperidoneAn atypical antipsychotic used in the treatment of schizophrenia and other schizoaffective or delusional disorders.
DrugDrug NameTargetType
DB09128BrexpiprazoleCytochrome P450 2D6enzyme
DB09128BrexpiprazoleCytochrome P450 3A4enzyme
DB09128Brexpiprazole5-hydroxytryptamine receptor 1Atarget
DB09128BrexpiprazoleDopamine D2 receptortarget
DB09128Brexpiprazole5-hydroxytryptamine receptor 2Atarget
DB09128BrexpiprazoleAlpha-2C adrenergic receptortarget
DB09128BrexpiprazoleAlpha-1B adrenergic receptortarget
DB09128BrexpiprazoleMultidrug and toxin extrusion protein 2transporter
DB09128BrexpiprazoleSerum albumincarrier
DB09128BrexpiprazoleAlpha-1-acid glycoprotein 1carrier
DB09128BrexpiprazoleDopamine D3 receptortarget
DB09128Brexpiprazole5-hydroxytryptamine receptor 2Btarget
DB09128Brexpiprazole5-hydroxytryptamine receptor 7target
DB09128BrexpiprazoleAlpha-1A adrenergic receptortarget
DB09128BrexpiprazoleAlpha-1D adrenergic receptortarget
DB09128BrexpiprazoleHistamine H1 receptortarget
DB09128BrexpiprazoleMuscarinic acetylcholine receptor M1target
DB01267PaliperidoneDopamine D2 receptortarget
DB01267Paliperidone5-hydroxytryptamine receptor 2Atarget
DB01267PaliperidoneHistamine H1 receptortarget
DB01267PaliperidoneAlpha-1A adrenergic receptortarget
DB01267PaliperidoneAlpha-1B adrenergic receptortarget
DB01267PaliperidoneDopamine D3 receptortarget
DB01267PaliperidoneDopamine D4 receptortarget
DB01267PaliperidoneDopamine D1 receptortarget
DB01267PaliperidoneAlpha-2A adrenergic receptortarget
DB01267PaliperidoneAlpha-2B adrenergic receptortarget
DB01267PaliperidoneAlpha-2C adrenergic receptortarget
DB01267Paliperidone5-hydroxytryptamine receptor 1Atarget
DB01267Paliperidone5-hydroxytryptamine receptor 1Dtarget
DB01267Paliperidone5-hydroxytryptamine receptor 2Ctarget
DB01267Paliperidone5-hydroxytryptamine receptor 7target
DB01267PaliperidoneCytochrome P450 3A4enzyme
DB01267PaliperidoneCytochrome P450 2D6enzyme
DB01267PaliperidoneCytochrome P450 3A5enzyme
DB01267PaliperidoneP-glycoprotein 1transporter
DrugDrug NamePhaseStatusCount
DB00472Fluoxetine4Unknown Status1
DB01017Minocycline4Completed1
DB00285Venlafaxine4Unknown Status1
DB00215CitalopramNot AvailableCompleted1
DB00215CitalopramNot AvailableUnknown Status2
DB01175EscitalopramNot AvailableCompleted1
DB00370MirtazapineNot AvailableCompleted1
DB06480PrucaloprideNot AvailableCompleted2
DB01104SertralineNot AvailableCompleted1
DB00285VenlafaxineNot AvailableCompleted1