OHT - Ocular Hypertension

Also known as: Ocular Hypertension / Ocular Hypertension (OH) / Hypertension Ocular / Ocular Hypertension (OHT) / Intraocular pressure high / Hypertension, Ocular / Ocular Hypertensive / Intraocular hypertension / Intra Ocular Hypertension / Ocular hypertension (disorder) / Intraocular pressure increased / Intraocular pressure raised / Raised intraocular pressure (finding) / IOP increased / Raised IOP / Ocular tension increased / Tension ocular increased / Pressure intraocular increased / Increased intraocular pressure

DrugDrug NameDrug Description
DB00964ApraclonidineAn alpha adrenergic agonist used to treat raised intraocular pressure.
DB00195BetaxololA cardioselective beta blocking agent commonly used to treat hypertension and elevated intraocular pressure (when administered ophthalmically).
DB00905BimatoprostA prostaglandin analog used to treat hypotrichosis of the eyelashes and intraocular pressure in open angle glaucoma or ocular hypertension.
DB00484BrimonidineAn alpha-2 adrenergic agonist used to treat glaucoma and ocular hypertension, as well as facial erythema in rosacea.
DB01194BrinzolamideA carbonic anhydrase inhibitor used for the reduction of elevated intraocular pressure in patients with ocular hypertension or open-angle glaucoma.
DB00521CarteololA beta adrenergic antagonist used to treat arrhythmia, angina, hypertension, and glaucoma.
DB00869DorzolamideA carbonic anhydrase inhibitor used to treat high intraocular pressure in ocular hypertension and open angle glaucoma.
DB09462GlycerinIt is used as a solvent, emollient, pharmaceutical agent, and sweetening agent.
DB00654LatanoprostAn isopropyl ester prodrug used to treat increased intraocular pressure.
DB01210LevobunololA beta-adrenergic antagonist used for the reduction of elevated intraocular pressure in patients with ocular hypertension or open-angle glaucoma.
DB01214MetipranololA beta-adrenergic antagonist used for the reduction of elevated intraocular pressure in patients with ocular hypertension or open-angle glaucoma.
DB13931NetarsudilA rho kinase inhibitor used to reduce intraocular pressure in patients with open angle glaucoma or ocular hypertension.
DB15071Omidenepag isopropylAn agonist of the prostaglandin EP2 receptor indicated for the reduction of elevated intraocular pressure.
DB01085PilocarpineA muscarinic agonist used to treat dry mouth and various ophthalmic conditions, such as presbyopia, increased intraocular pressure, and angle-closure glaucoma.
DB13165RipasudilA rho kinase inhibitor indicated to treat ocular hypertension and open-angle glaucoma.
DB08819TafluprostAn ophthalmic prostaglandin analog used to lower intraocular pressure in patients with ocular hypertension or open-angle glaucoma.
DB00373TimololA non-selective beta adrenergic blocker used in the treatment of elevated intraocular pressure in ocular hypertension or open angle glaucoma.
DB00287TravoprostA prostaglandin analog used in the treatment of elevated intraocular pressure due to open angle glaucoma or ocular hypertension.
DB06826UnoprostoneA prostaglandin analogue used to lower intraocular pressure in patients with open-angle glaucoma or ocular hypertension who are clinically unresponsive to other ocular antihypertensive agents.
DrugDrug NameTargetType
DB00964ApraclonidineAlpha-2A adrenergic receptortarget
DB00964ApraclonidineAlpha-1A adrenergic receptortarget
DB00964ApraclonidineAlpha-2B adrenergic receptortarget
DB00195BetaxololBeta-1 adrenergic receptortarget
DB00195BetaxololBeta-2 adrenergic receptortarget
DB00195BetaxololCytochrome P450 1A2enzyme
DB00195BetaxololCytochrome P450 2D6enzyme
DB00905BimatoprostProstaglandin F2-alpha receptortarget
DB00905BimatoprostProstaglandin E2 receptor EP1 subtypetarget
DB00905BimatoprostProstaglandin E2 receptor EP3 subtypetarget
DB00905BimatoprostCytochrome P450 3A4enzyme
DB00905BimatoprostCytochrome P450 3A5enzyme
DB00484BrimonidineAlpha-2A adrenergic receptortarget
DB00484BrimonidineAlpha-2B adrenergic receptortarget
DB00484BrimonidineAlpha-2C adrenergic receptortarget
DB00484BrimonidineAldehyde oxidaseenzyme
DB01194BrinzolamideCarbonic anhydrase 1target
DB01194BrinzolamideCarbonic anhydrase 2target
DB01194BrinzolamideCytochrome P450 3A4enzyme
DB01194BrinzolamideCarbonic anhydrase 5A, mitochondrialtarget
DB01194BrinzolamideCarbonic anhydrase 4target
DB01194BrinzolamideCarbonic anhydrase 3target
DB01194BrinzolamideCytochrome P450 2A6enzyme
DB01194BrinzolamideCytochrome P450 2B6enzyme
DB01194BrinzolamideCytochrome P450 2C8enzyme
DB01194BrinzolamideCytochrome P450 2C9enzyme
DB00521CarteololBeta-2 adrenergic receptortarget
DB00521CarteololBeta-1 adrenergic receptortarget
DB00521CarteololCytochrome P450 2D6enzyme
DB00869DorzolamideCarbonic anhydrase 2target
DB00869DorzolamideCarbonic anhydrase 1target
DB00869DorzolamideCarbonic anhydrase 4target
DB00869DorzolamideCytochrome P450 2C9enzyme
DB00869DorzolamideCarbonic anhydrase 3target
DB00869DorzolamideCytochrome P450 2B1enzyme
DB00869DorzolamideCytochrome P450 2E1enzyme
DB00869DorzolamideCytochrome P450 3A2enzyme
DB09462GlycerinGroup IIE secretory phospholipase A2target
DB09462GlycerinInositol-3-phosphate synthase 1target
DB09462GlycerinAlcohol dehydrogenase 1Btarget
DB09462GlycerinInositol 1,4,5-trisphosphate receptor type 1target
DB09462GlycerinGlycodelintarget
DB09462GlycerinAlpha-N-acetylgalactosaminidasetarget
DB09462GlycerinADP-ribosylation factor 1target
DB09462GlycerinBifunctional 3'-phosphoadenosine 5'-phosphosulfate synthase 1target
DB09462GlycerinDNA mismatch repair protein MutLtarget
DB09462GlycerinRibonucleoside-diphosphate reductase 1 subunit betatarget
DB09462GlycerinA/G-specific adenine glycosylasetarget
DB09462GlycerintRNA (cytosine(38)-C(5))-methyltransferasetarget
DB09462GlycerinCytochrome P450 2E1enzyme
DB09462GlycerinRetinal dehydrogenase 1enzyme
DB09462GlycerinPeroxisome proliferator-activated receptor deltatarget
DB09462GlycerinMaleylacetoacetate isomerasetarget
DB09462GlycerinAquaporin-7transporter
DB09462GlycerinAquaporin-9transporter
DB09462GlycerinGlycerol uptake facilitator proteintransporter
DB00654LatanoprostProstaglandin F2-alpha receptortarget
DB00654LatanoprostSolute carrier organic anion transporter family member 2A1transporter
DB00654LatanoprostSolute carrier family 22 member 6transporter
DB00654LatanoprostSolute carrier family 22 member 8transporter
DB00654LatanoprostCorneal esterasesenzyme
DB01210LevobunololBeta-1 adrenergic receptortarget
DB01210LevobunololBeta-2 adrenergic receptortarget
DB01210LevobunololCytochrome P450 2D6enzyme
DB01214MetipranololBeta-1 adrenergic receptortarget
DB01214MetipranololBeta-2 adrenergic receptortarget
DB01214MetipranololCytochrome P450 2D6enzyme
DB13931NetarsudilRho-associated protein kinase 1target
DB13931NetarsudilRho-associated protein kinase 2target
DB13931NetarsudilSodium-dependent noradrenaline transportertarget
DB15071Omidenepag isopropylCarboxylesteraseenzyme
DB15071Omidenepag isopropylProstaglandin E2 receptor EP2 subtypetarget
DB15071Omidenepag isopropylProstaglandin E2 receptor EP1 subtypetarget
DB01085PilocarpineMuscarinic acetylcholine receptor M1target
DB01085PilocarpineMuscarinic acetylcholine receptor M2target
DB01085PilocarpineCytochrome P450 2A6enzyme
DB01085PilocarpineMuscarinic acetylcholine receptor M3target
DB01085PilocarpineCytochrome P450 3A4enzyme
DB01085PilocarpineMuscarinic acetylcholine receptor M4target
DB01085PilocarpineMuscarinic acetylcholine receptor M5target
DB01085PilocarpineSerum paraoxonase/arylesterase 1enzyme
DB13165RipasudilRho-associated protein kinase 1target
DB13165RipasudilRho-associated protein kinase 2target
DB08819TafluprostProstaglandin F2-alpha receptortarget
DB08819TafluprostProstaglandin G/H synthase 2enzyme
DB00373TimololBeta-1 adrenergic receptortarget
DB00373TimololBeta-2 adrenergic receptortarget
DB00373TimololCytochrome P450 2D6enzyme
DB00373TimololP-glycoprotein 1transporter
DB00373TimololCytochrome P450 2C19enzyme
DB00373TimololLysozymetarget
DB00287TravoprostProstaglandin F2-alpha receptortarget
DrugDrug NamePhaseStatusCount
DB12256Bamosiran1Completed1
DB00905Bimatoprost1Not Yet Recruiting1
DB00484Brimonidine1Completed1
DB00521Carteolol1Completed1
DB00869Dorzolamide1Completed1
DB00654Latanoprost1Completed3
DB00654Latanoprost1Recruiting2
DB00654Latanoprost1Terminated1
DB16353Razuprotafib1Completed1
DB18614ST2661Completed1
DB12043Sepetaprost1Completed1
DB08819Tafluprost1Completed1
DB00373Timolol1Completed2
DB00287Travoprost1Completed1
DB12256Bamosiran1 / 2Completed1
DB00905Bimatoprost1 / 2Completed3
DB00905Bimatoprost1 / 2Recruiting1
DB05757DNB-0011 / 2Completed1
DB12116Epigallocatechin gallate1 / 2Unknown Status1
DB12295Evodenoson1 / 2Completed1
DB16009LX-71011 / 2Completed1
DB00654Latanoprost1 / 2Active Not Recruiting1
DB00654Latanoprost1 / 2Completed5
DB16112OT-7301 / 2Completed1
DB12977Simenepag isopropyl1 / 2Completed1
DB00373Timolol1 / 2Completed4
DB00373Timolol1 / 2Recruiting1
DB00373Timolol1 / 2Unknown Status1
DB13122Trabodenoson1 / 2Completed1
DB16085Aganepag isopropyl2Completed1
DB13906Aloe vera leaf2Completed1
DB05288Anecortave acetate2Terminated1
DB12256Bamosiran2Completed2
DB11105Benzalkonium2Completed1
DB00905Bimatoprost2Active Not Recruiting1
DB00905Bimatoprost2Completed12
DB00484Brimonidine2Completed4
DB00484Brimonidine2Terminated1
DB01194Brinzolamide2Completed4
DB01194Brinzolamide2Terminated1
DB14322Coconut oil2Completed1
DB00869Dorzolamide2Completed1
DB00869Dorzolamide2Not Yet Recruiting1
DB00869Dorzolamide2Unknown Status1
DB08818Hyaluronic acid2Completed1
DB00654Latanoprost2Completed32
DB00654Latanoprost2Unknown Status2
DB00654Latanoprost2Withdrawn2
DB11660Latanoprostene bunod2Completed1
DB04861Nebivolol2Completed1
DB13931Netarsudil2Completed5
DB15071Omidenepag isopropyl2Completed1
DB05746PF-031872072Completed2
DB00692Phentolamine2Completed1
DB05511Piclidenoson2Completed1
DB01839Propylene glycol2Completed1
DB16353Razuprotafib2Completed1
DB14272Rosemary2Completed1
DB06195Seliciclib2Completed1
DB12043Sepetaprost2Completed1
DB12977Simenepag isopropyl2Completed2
DB12623Taprenepag2Completed2
DB00373Timolol2Completed16
DB00373Timolol2Not Yet Recruiting1
DB00373Timolol2Recruiting2
DB13122Trabodenoson2Completed2
DB00287Travoprost2Active Not Recruiting1
DB00287Travoprost2Completed10
DB00287Travoprost2Recruiting1
DB00287Travoprost2Terminated1
DB00905Bimatoprost2 / 3Completed1
DB00654Latanoprost2 / 3Completed1
DB15071Omidenepag isopropyl2 / 3Completed1
DB00195Betaxolol3Completed3
DB00905Bimatoprost3Active Not Recruiting1
DB00905Bimatoprost3Completed17
DB00905Bimatoprost3Enrolling by Invitation1
DB00905Bimatoprost3Recruiting1
DB00905Bimatoprost3Withdrawn1
DB00484Brimonidine3Completed19
DB00484Brimonidine3Withdrawn1
DB01194Brinzolamide3Completed12
DB01194Brinzolamide3Terminated2
DB01194Brinzolamide3Withdrawn1
DB00521Carteolol3Completed1
DB00869Dorzolamide3Completed7
DB00869Dorzolamide3Terminated1
DB00869Dorzolamide3Withdrawn1
DB00654Latanoprost3Completed29
DB00654Latanoprost3Recruiting1
DB00654Latanoprost3Terminated2
DB00654Latanoprost3Unknown Status1
DB00654Latanoprost3Withdrawn2
DB11660Latanoprostene bunod3Completed3
DB09351Levobetaxolol3Completed2
DB13931Netarsudil3Completed8
DB01165Ofloxacin3Withdrawn1
DB01085Pilocarpine3Withdrawn1
DB00860Prednisolone3Withdrawn1
DB13165Ripasudil3Completed1
DB08819Tafluprost3Completed7
DB00373Timolol3Completed58
DB00373Timolol3Terminated2
DB00373Timolol3Withdrawn2
DB13122Trabodenoson3Completed1
DB00287Travoprost3Active Not Recruiting2
DB00287Travoprost3Completed21
DB00287Travoprost3Recruiting1
DB00287Travoprost3Terminated3
DB00287Travoprost3Withdrawn2
DB00905Bimatoprost4Completed27
DB00905Bimatoprost4Unknown Status1
DB00905Bimatoprost4Withdrawn1
DB00484Brimonidine4Completed18
DB00484Brimonidine4Terminated2
DB00484Brimonidine4Unknown Status1
DB01194Brinzolamide4Completed17
DB01194Brinzolamide4Terminated1
DB01234Dexamethasone4Completed1
DB01075Diphenhydramine4Completed2
DB00869Dorzolamide4Completed14
DB00869Dorzolamide4Recruiting1
DB00869Dorzolamide4Terminated2
DB11114Eucalyptus oil4Completed1
DB00588Fluticasone propionate4Completed1
DB11075Hypromellose4Completed4
DB16956L-Acetylleucine4Completed1
DB16956L-Acetylleucine4Terminated1
DB00654Latanoprost4Completed30
DB00654Latanoprost4Recruiting3
DB00654Latanoprost4Terminated2
DB00654Latanoprost4Unknown Status1
DB00654Latanoprost4Withdrawn1
DB11660Latanoprostene bunod4Withdrawn1
DB14596Loteprednol etabonate4Completed1
DB01043Memantine4Completed1
DB13931Netarsudil4Completed1
DB15071Omidenepag isopropyl4Recruiting1
DB10984Peppermint4Completed1
DB11077Polyethylene glycol 4004Completed1
DB00860Prednisolone4Unknown Status1
DB01839Propylene glycol4Completed1
DB08819Tafluprost4Completed6
DB08819Tafluprost4Recruiting1
DB08819Tafluprost4Unknown Status1
DB08819Tafluprost4Withdrawn1
DB00373Timolol4Completed36
DB00373Timolol4Recruiting3
DB00373Timolol4Terminated3
DB00373Timolol4Withdrawn3
DB00684Tobramycin4Completed1
DB00287Travoprost4Completed31
DB00287Travoprost4Terminated2
DB00287Travoprost4Withdrawn3
DB11195Xylitol4Completed1
DB00964ApraclonidineNot AvailableUnknown Status1
DB00905BimatoprostNot AvailableCompleted14
DB00905BimatoprostNot AvailableUnknown Status1
DB00484BrimonidineNot AvailableCompleted4
DB00484BrimonidineNot AvailableUnknown Status1
DB00484BrimonidineNot AvailableWithdrawn1
DB01194BrinzolamideNot AvailableCompleted1
DB01194BrinzolamideNot AvailableUnknown Status1
DB00869DorzolamideNot AvailableUnknown Status1
DB00869DorzolamideNot AvailableWithdrawn1
DB01050IbuprofenNot AvailableCompleted1
DB00654LatanoprostNot AvailableCompleted6
DB00654LatanoprostNot AvailableRecruiting1
DB00654LatanoprostNot AvailableUnknown Status5
DB00654LatanoprostNot AvailableWithdrawn1
DB11660Latanoprostene bunodNot AvailableCompleted1
DB14596Loteprednol etabonateNot AvailableCompleted1
DB13931NetarsudilNot AvailableCompleted1
DB01085PilocarpineNot AvailableCompleted1
DB01085PilocarpineNot AvailableUnknown Status1
DB15566Prednisolone acetateNot AvailableNot Yet Recruiting1
DB00373TimololNot AvailableCompleted13
DB00373TimololNot AvailableRecruiting1
DB00373TimololNot AvailableUnknown Status1
DB00373TimololNot AvailableWithdrawn2
DB00684TobramycinNot AvailableCompleted1
DB00287TravoprostNot AvailableCompleted6
DB00287TravoprostNot AvailableTerminated1
DB00287TravoprostNot AvailableUnknown Status1
DB00620TriamcinoloneNot AvailableNot Yet Recruiting1