Metastatic RET-fusion Non Small Cell Lung Cancer

DrugDrug NameDrug Description
DB15822PralsetinibA RET receptor tyrosine kinase inhibitor for the treatment of metastatic RET-driven non-small cell lung cancer.
DB15685SelpercatinibA RET receptor tyrosine kinase inhibitor for the treatment of RET-driven non-small cell lung cancer, medullary thyroid cancer, and thyroid cancer in appropriate patient populations.
DrugDrug NameTargetType
DB15822PralsetinibProto-oncogene tyrosine-protein kinase receptor Rettarget
DB15822PralsetinibEpithelial discoidin domain-containing receptor 1target
DB15822PralsetinibNT-3 growth factor receptortarget
DB15822PralsetinibReceptor-type tyrosine-protein kinase FLT3target
DB15822PralsetinibTyrosine-protein kinase JAK1target
DB15822PralsetinibTyrosine-protein kinase JAK2target
DB15822PralsetinibHigh affinity nerve growth factor receptortarget
DB15822PralsetinibVascular endothelial growth factor receptor 2target
DB15822PralsetinibPlatelet-derived growth factor receptor betatarget
DB15822PralsetinibFibroblast growth factor receptor 1target
DB15822PralsetinibFibroblast growth factor receptor 2target
DB15822PralsetinibCytochrome P450 3A4enzyme
DB15822PralsetinibCytochrome P450 3A5enzyme
DB15822PralsetinibCytochrome P450 2D6enzyme
DB15822PralsetinibCytochrome P450 1A2enzyme
DB15822PralsetinibCytochrome P450 2C8enzyme
DB15822PralsetinibCytochrome P450 2C9enzyme
DB15822PralsetinibP-glycoprotein 1transporter
DB15822PralsetinibATP-binding cassette sub-family G member 2transporter
DB15822PralsetinibSolute carrier organic anion transporter family member 1B1transporter
DB15822PralsetinibSolute carrier organic anion transporter family member 1B3transporter
DB15822PralsetinibSolute carrier family 22 member 6transporter
DB15822PralsetinibMultidrug and toxin extrusion protein 1transporter
DB15822PralsetinibMultidrug and toxin extrusion protein 2transporter
DB15822PralsetinibBile salt export pumptransporter
DB15685SelpercatinibProto-oncogene tyrosine-protein kinase receptor Rettarget
DB15685SelpercatinibVascular endothelial growth factor receptor 1target
DB15685SelpercatinibVascular endothelial growth factor receptor 3target
DB15685SelpercatinibFibroblast growth factor receptor 1target
DB15685SelpercatinibFibroblast growth factor receptor 2target
DB15685SelpercatinibFibroblast growth factor receptor 3target
DB15685SelpercatinibCytochrome P450 3A4enzyme
DB15685SelpercatinibCytochrome P450 2C8enzyme
DB15685SelpercatinibCytochrome P450 3A Subfamilyenzyme
DB15685SelpercatinibP-glycoprotein 1transporter
DB15685SelpercatinibATP-binding cassette sub-family G member 2transporter
DB15685SelpercatinibMultidrug and toxin extrusion protein 1transporter
DrugDrug NamePhaseStatusCount