| Pralsetinib | transporter | Multidrug and toxin extrusion protein 1 | Details |
| Pralsetinib | transporter | Bile salt export pump | Details |
| Copper oxodotreotide Cu-64 | target | Somatostatin receptor type 2 | Details |
| Agalsidase alfa | target | Globotriaosylceramide | Details |
| Agalsidase alfa | transporter | Cation-dependent mannose-6-phosphate receptor | Details |
| Etesevimab | target | Spike glycoprotein | Details |
| Atoltivimab | target | Envelope glycoprotein | Details |
| Maftivimab | target | Envelope glycoprotein | Details |
| Odesivimab | target | Envelope glycoprotein | Details |
| Lumasiran | target | Hydroxyacid oxidase 1 | Details |
| Lumasiran | carrier | Serum albumin | Details |
| Lumasiran | enzyme | Cytochrome P450 2C8 | Details |
| Imdevimab | target | Spike glycoprotein | Details |
| Casirivimab | target | Spike glycoprotein | Details |
| Naxitamab | target | GD2 disialoganglioside | Details |
| Berotralstat | enzyme | Cytochrome P450 2D6 | Details |
| Berotralstat | transporter | ATP-binding cassette sub-family G member 2 | Details |
| Berotralstat | target | Plasma kallikrein | Details |
| Berotralstat | enzyme | Cytochrome P450 3A4 | Details |
| Berotralstat | transporter | P-glycoprotein 1 | Details |
| Gallium Ga-68 gozetotide | target | Prostate-specific antigen | Details |
| Razuprotafib | target | Receptor-type tyrosine-protein phosphatase beta | Details |
| Mezagitamab | target | ADP-ribosyl cyclase 1 | Details |
| Ansuvimab | target | Envelope glycoprotein | Details |