| Tilsotolimod | target | Toll-like receptor 9 | Details |
| Tropifexor | target | Bile acid receptor | Details |
| Veliflapon | target | Arachidonate 5-lipoxygenase-activating protein | Details |
| Vicagrel | enzyme | Cytochrome P450 2C19 | Details |
| Vicagrel | enzyme | Cocaine esterase | Details |
| Vicagrel | enzyme | Intestinal-type alkaline phosphatase | Details |
| Vicagrel | target | P2Y purinoceptor 12 | Details |
| Vicagrel | enzyme | Arylacetamide deacetylase | Details |
| Vicagrel | enzyme | Liver carboxylesterase 1 | Details |
| Volinanserin | target | 5-hydroxytryptamine receptor 2A | Details |
| Razuprotafib | target | Receptor-type tyrosine-protein phosphatase beta | Details |
| Sotrovimab | target | Spike glycoprotein | Details |
| Mezagitamab | target | ADP-ribosyl cyclase 1 | Details |
| Garetosmab | target | Inhibin beta A chain | Details |
| Ansuvimab | target | Envelope glycoprotein | Details |
| Mobocertinib | transporter | ATP-binding cassette sub-family G member 2 | Details |
| Mobocertinib | enzyme | Cytochrome P450 3A4 | Details |
| Mobocertinib | target | Epidermal growth factor receptor | Details |
| Mobocertinib | enzyme | Cytochrome P450 3A5 | Details |
| Mobocertinib | enzyme | Cytochrome P450 3A7 | Details |
| Mobocertinib | transporter | P-glycoprotein 1 | Details |
| Cilgavimab | target | Spike glycoprotein | Details |
| Tixagevimab | target | Spike glycoprotein | Details |
| Regdanvimab | target | Spike glycoprotein | Details |
| Azvudine | target | Canalicular multispecific organic anion transporter 1 | Details |
| Azvudine | target | ATP-binding cassette sub-family G member 2 | Details |
| Azvudine | target | P-glycoprotein 1 | Details |
| Camidanlumab tesirine | target | Interleukin-2 receptor subunit alpha | Details |
| Vilobelimab | target | Complement C5 | Details |
| Geptanolimab | target | Programmed cell death protein 1 | Details |