| Prolgolimab | target | Programmed cell death protein 1 | Details |
| TPMPA | target | Gamma-aminobutyric acid receptor subunit rho-1 | Details |
| TPMPA | target | Gamma-aminobutyric acid receptor subunit rho-3 | Details |
| TPMPA | target | Gamma-aminobutyric acid receptor subunit rho-2 | Details |
| Bebtelovimab | target | Spike glycoprotein | Details |
| Ivarmacitinib | target | Tyrosine-protein kinase JAK1 | Details |
| Lutetium Lu-177 vipivotide tetraxetan | target | Prostate-specific antigen | Details |
| Letibotulinumtoxina | target | Synaptosomal-associated protein 25 | Details |
| Indigo | target | Aryl hydrocarbon receptor | Details |
| Betibeglogene autotemcel | target | Alpha globin | Details |
| KW-6356 | target | Adenosine receptor A2a | Details |
| Linzagolix | target | Gonadotropin-releasing hormone receptor | Details |
| Linzagolix | transporter | Solute carrier organic anion transporter family member 1B3 | Details |
| Linzagolix | transporter | ATP-binding cassette sub-family G member 2 | Details |
| Linzagolix | transporter | Solute carrier family 22 member 6 | Details |
| Linzagolix | enzyme | Cytochrome P450 3A4 | Details |
| Linzagolix | transporter | Solute carrier organic anion transporter family member 1B1 | Details |
| Linzagolix | enzyme | Cytochrome P450 2C8 | Details |
| Linzagolix | carrier | Serum albumin | Details |
| Linzagolix | enzyme | Cytochrome P450 2C9 | Details |
| Linzagolix | transporter | Solute carrier family 22 member 8 | Details |
| JNJ-17216498 | target | Histamine H3 receptor | Details |
| UCB7362 | target | Plasmepsin X | Details |
| UCB7362 | target | Plasmepsin X | Details |
| Anacaulase | enzyme | Cytochrome P450 2C9 | Details |
| Anacaulase | enzyme | Cytochrome P450 2C8 | Details |
| Anacaulase | target | Alpha-1-antichymotrypsin | Details |
| Anacaulase | target | Alpha-2-macroglobulin | Details |