| DB00304 | Desogestrel | approved | yes | agonist | Details |
| DB00351 | Megestrol acetate | approved, investigational, vet_approved | yes | agonist | Details |
| DB00367 | Levonorgestrel | approved, investigational | yes | modulator | Details |
| DB00378 | Dydrogesterone | approved, investigational, withdrawn | yes | agonist | Details |
| DB00396 | Progesterone | approved, vet_approved | yes | agonist | Details |
| DB00603 | Medroxyprogesterone acetate | approved, investigational | yes | agonist | Details |
| DB00717 | Norethisterone | approved | yes | agonist | Details |
| DB00834 | Mifepristone | approved, investigational | yes | antagonist | Details |
| DB00957 | Norgestimate | approved, investigational | yes | agonist | Details |
| DB00294 | Etonogestrel | approved, investigational | yes | agonist | Details |
| DB00823 | Ethynodiol diacetate | approved | yes | agonist | Details |
| DB01395 | Drospirenone | approved | yes | agonist | Details |
| DB02998 | Metribolone | experimental | unknown | | Details |
| DB05253 | Telapristone acetate | investigational | unknown | | Details |
| DB04787 | Tanaproget | investigational | yes | agonist | Details |
| DB06680 | Asoprisnil | investigational | unknown | | Details |
| DB01406 | Danazol | approved | yes | agonist | Details |
| DB01431 | Allylestrenol | experimental | yes | agonist | Details |
| DB00588 | Fluticasone propionate | approved | unknown | agonist | Details |
| DB06713 | Norelgestromin | approved, investigational | yes | agonist | Details |
| DB08867 | Ulipristal | approved | yes | modulator | Details |
| DB00421 | Spironolactone | approved | unknown | agonist | Details |
| DB06789 | Hydroxyprogesterone caproate | approved, investigational | unknown | agonist | Details |
| DB09389 | Norgestrel | approved | yes | binder | Details |
| DB00431 | Lindane | approved, withdrawn | unknown | | Details |
| DB00648 | Mitotane | approved | unknown | | Details |
| DB02746 | Phthalic Acid | experimental | unknown | | Details |
| DB00764 | Mometasone | experimental | unknown | agonist | Details |
| DB11219 | Enzacamene | approved | unknown | antagonist | Details |
| DB11064 | Homosalate | approved, investigational | unknown | antagonist | Details |
| DB01428 | Oxybenzone | approved, investigational | unknown | antagonist | Details |
| DB06730 | Gestodene | investigational | yes | binderactivator | Details |
| DB09123 | Dienogest | approved | yes | agonist | Details |
| DB09124 | Medrogestone | approved, withdrawn | yes | ligand | Details |
| DB11619 | Gestrinone | approved | unknown | antagonistagonist | Details |
| DB13857 | Demegestone | experimental | yes | agonist | Details |
| DB14512 | Mometasone furoate | approved, investigational, vet_approved | unknown | | Details |
| DB14583 | Segesterone acetate | approved, experimental, investigational | yes | agonistactivator | Details |
| DB13867 | Fluticasone | approved, experimental | unknown | agonist | Details |
| DB08906 | Fluticasone furoate | approved | unknown | agonist | Details |
| DB12941 | Darolutamide | approved, investigational | unknown | antagonist | Details |