| Lepirudin | target | Prothrombin | Details |
| Cetuximab | target | Epidermal growth factor receptor | Details |
| Cetuximab | target | Low affinity immunoglobulin gamma Fc region receptor III-B | Details |
| Cetuximab | target | Low affinity immunoglobulin gamma Fc region receptor III-A | Details |
| Cetuximab | target | Complement C1q subcomponent subunit A | Details |
| Cetuximab | target | Complement C1q subcomponent subunit B | Details |
| Cetuximab | target | Complement C1q subcomponent subunit C | Details |
| Cetuximab | target | High affinity immunoglobulin gamma Fc receptor I | Details |
| Cetuximab | target | Low affinity immunoglobulin gamma Fc region receptor II-a | Details |
| Dornase alfa | target | DNA | Details |
| Denileukin diftitox | target | Interleukin-2 receptor subunit alpha | Details |
| Denileukin diftitox | target | Cytokine receptor common subunit gamma | Details |
| Denileukin diftitox | target | Interleukin-2 receptor subunit beta | Details |
| Etanercept | target | Tumor necrosis factor | Details |
| Etanercept | target | Low affinity immunoglobulin gamma Fc region receptor III-A | Details |
| Etanercept | target | Complement component 1q (C1q) | Details |
| Etanercept | target | Lymphotoxin-alpha | Details |
| Etanercept | target | Low affinity immunoglobulin gamma Fc region receptor III-B | Details |
| Etanercept | target | High affinity immunoglobulin gamma Fc receptor I | Details |
| Etanercept | target | Low affinity immunoglobulin gamma Fc region receptor II-a | Details |
| Etanercept | target | Low affinity immunoglobulin gamma Fc region receptor II-b | Details |
| Etanercept | target | Low affinity immunoglobulin gamma Fc region receptor II-c | Details |
| Bivalirudin | target | Prothrombin | Details |
| Bivalirudin | enzyme | Myeloperoxidase | Details |
| Leuprolide | target | Gonadotropin-releasing hormone receptor | Details |
| Peginterferon alfa-2a | target | Interferon alpha/beta receptor 2 | Details |
| Peginterferon alfa-2a | target | Interferon alpha/beta receptor 1 | Details |
| Peginterferon alfa-2a | enzyme | Cytochrome P450 1A2 | Details |
| Alteplase | target | Plasminogen activator inhibitor 1 | Details |
| Alteplase | target | Plasminogen | Details |