Gastrin/cholecystokinin type B receptor

BE0001158ProteinHumansCCKBR

Receptor for the peptide hormones gastrin and cholecystokinin (CCK). It is acted on by 13 drugs in DrugBank.

Gene name
CCKBR
UniProtKB entry
P32239Swiss-Prot
Cellular location
Cell membrane
Residues / weight
447 residues · 48,419 Da
Also known as
CCK-B receptor · CCK-BR · CCK2-R · CCKRB · Cholecystokinin-2 receptor

Resolves to

Protein
UniProtP32239UniProt nameGASR_HUMAN
Gene
HGNCHGNC:1571NCBI Gene887GenBank306489GeneCardsCCKBR
Pharmacology
IUPHAR/GtoPdb77KEGGhsa:887
Structure
PDB1L4TPDB7F8VPDB7F8W
Drugs

What you can answer from here — as of September 07, 2019

13DrugsApproved to experimental, with action, bond type and pharmacological action
Sign in
4GO termsFunction, process and component, as structured annotations
Sign in
1Pfam domainDomain architecture mapped to Pfam families and clans
Sign in
54+ReferencesStructured and connected to the statements they support
Sign in

Which approved drugs act on Gastrin/cholecystokinin type B receptor, how selective are they, and which programs against it are still in active trials?

Answer this in Biopharma OSSign in to your account

Create a free account or log in to explore the full data card.

Create Account
Log InPaid Account Log In