| DB00601 | Linezolid | approved, investigational | yes | inhibitor | Details |
| DB00954 | Dirithromycin | experimental | yes | inhibitor | Details |
| DB00976 | Telithromycin | approved | yes | inhibitor | Details |
| DB04850 | Posizolid | investigational | yes | antagonistblocker | Details |
| DB00207 | Azithromycin | approved | yes | inhibitor | Details |
| DB00199 | Erythromycin | approved, investigational, vet_approved | yes | inhibitor | Details |
| DB06419 | Cethromycin | investigational | yes | antagonist | Details |
| DB01369 | Quinupristin | approved | yes | inhibitor | Details |
| DB14569 | Tedizolid | approved, investigational | yes | inhibitor | Details |
| DB09042 | Tedizolid phosphate | approved | yes | inhibitor | Details |
| DB00684 | Tobramycin | approved, investigational | yes | inhibitor | Details |
| DB01082 | Streptomycin | approved, vet_approved | yes | inhibitor | Details |
| DB01627 | Lincomycin | approved, vet_approved | yes | binder | Details |
| DB00798 | Gentamicin | approved, vet_approved | yes | inhibitor | Details |