Gastrin-releasing peptide receptor

BE0012984ProteinHumansGRPR

Receptor for gastrin-releasing peptide (GRP) (PubMed:1655761). It is acted on by 3 drugs in DrugBank.

Gene name
GRPR
UniProtKB entry
P30550Swiss-Prot
Cellular location
Cell membrane
Residues / weight
384 residues · 43,198 Da
Also known as
GRP-preferring bombesin receptor · GRP-R

Resolves to

Protein
UniProtP30550UniProt nameGRPR_HUMAN
Gene
HGNCHGNC:4609NCBI Gene2925GeneCardsGRPR
Pharmacology
IUPHAR/GtoPdb39KEGGhsa:2925
Structure
PDB7W3ZPDB7W40PDB7W41
Drugs

What you can answer from here — as of September 03, 2024

3DrugsApproved to experimental, with action, bond type and pharmacological action
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13GO termsFunction, process and component, as structured annotations
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1Pfam domainDomain architecture mapped to Pfam families and clans
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3+ReferencesStructured and connected to the statements they support
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Which compounds in development act on Gastrin-releasing peptide receptor, and which indications are they being tested in?

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