Excitatory Amino Acid Agonists

Name
Excitatory Amino Acid Agonists
Accession Number
DBCAT001301
Description

Drugs that bind to and activate excitatory amino acid receptors.

Drugs
DrugDrug Description
Quisqualic acidQuisqualic acid is an agonist at two subsets of excitatory amino acid receptors, ionotropic receptors that directly control membrane channels and metabotropic receptors that indirectly mediate calcium mobilization from intracellular...
KetamineA rapid-acting general anesthetic and NMDA receptor antagonist used for induction of anesthesia diagnostic and surgical procedures typically in combination with a muscle relaxant.
Drugs & Drug Targets
DrugTargetType
Quisqualic acidGlutamate receptor 2target
Quisqualic acidGlutamate receptor ionotropic, kainate 2target
KetamineGlutamate receptor ionotropic, NMDA 3Atarget
KetamineNeurokinin 1 receptortarget
KetamineCytochrome P450 2B6enzyme
KetamineCytochrome P450 2C9enzyme
KetamineCytochrome P450 3A4enzyme
KetamineDopamine D2 receptortarget
KetamineProstaglandin G/H synthase 1enzyme
KetamineCytochrome P450 2C8enzyme
KetamineDelta-type opioid receptortarget
KetamineSodium-dependent noradrenaline transportertarget
KetamineKappa-type opioid receptortarget
KetamineMu-type opioid receptortarget
KetamineMuscarinic acetylcholine receptortarget
Ketamine5-hydroxytryptamine receptor 2target
Ketamine5-hydroxytryptamine receptor 1target
Ketamine5-hydroxytryptamine receptor 3Atarget
KetamineNeuronal acetylcholine receptor subunit alpha-7target
KetamineCholinesterasetarget
KetamineNitric oxide synthase, braintarget