Antiandrogens, non-steroidal
- Name
- Antiandrogens, non-steroidal
- Accession Number
- DBCAT002767
- Description
Non steroidal compounds which inhibit or antagonize the biosynthesis or actions of androgens.
- Drugs
Drug Drug Description Flutamide An antiandrogen used for locally confined stage B2-C and D-2 metastatic prostate carcinoma. Nilutamide An antineoplastic hormone used to treat prostate cancer. Bicalutamide An androgen receptor inhibitor used to treat Stage D2 metastatic carcinoma of the prostate. Enzalutamide A second-generation androgen receptor inhibitor used to treat castration-resistant prostate cancer and metastatic castration-sensitive prostate cancer. Darolutamide An androgen receptor antagonist used for castration-resistant, non-metastatic prostate cancer and metastatic hormone-sensitive prostate cancer. Ketodarolutamide Ketodarolutamide, a nonsteroidal antiandrogen (NSAA), is the major active metabolite of darolutamide. - Drugs & Drug Targets