Receptors, Histamine H3

Name
Receptors, Histamine H3
Accession Number
DBCAT003022
Description

Not Available

Drugs
DrugDrug Description
PitolisantAn antagonist and inverse agonist at the histamine H3 receptor that is used to treat narcolepsy in adults.
IrdabisantIrdabisant has been used in trials studying Cognitive Impairment.
Drugs & Drug Targets
DrugTargetType
PitolisantHistamine H3 receptortarget
PitolisantCytochrome P450 3A4enzyme
PitolisantCytochrome P450 2D6enzyme
PitolisantCytochrome P450 1A2enzyme
PitolisantCytochrome P450 2B6enzyme
PitolisantSolute carrier family 22 member 1transporter
PitolisantPotassium voltage-gated channel subfamily H member 2target
PitolisantSerum albumincarrier
PitolisantAlpha-1-acid glycoprotein 1carrier