Tropomyosin Receptor Kinases Inhibitors

Name
Tropomyosin Receptor Kinases Inhibitors
Accession Number
DBCAT005471
Description

Not Available

Drugs
DrugDrug Description
LarotrectinibA kinase inhibitor used to treat solid tumors with neurotrophic receptor tyrosine kinase gene fusion, are metastatic, high risk for surgery, or have no alternative treatments.
Drugs & Drug Targets
DrugTargetType
LarotrectinibCytochrome P450 3A4enzyme
LarotrectinibHigh affinity nerve growth factor receptortarget
LarotrectinibBDNF/NT-3 growth factors receptortarget
LarotrectinibNT-3 growth factor receptortarget
LarotrectinibP-glycoprotein 1transporter
LarotrectinibATP-binding cassette sub-family G member 2transporter