Non-Competitive N-Methyl D-Aspartate (NMDA) Receptor Antagonists

Name
Non-Competitive N-Methyl D-Aspartate (NMDA) Receptor Antagonists
Accession Number
DBCAT005693
Description

Antagonists of NMDA receptors which exert their antagonism via binding to allosteric sites.

Drugs
DrugDrug Description
EsketamineA NMDA receptor antagonist used for treatment-resistant depression.
Drugs & Drug Targets
DrugTargetType
EsketamineNMDA receptortarget
EsketamineCytochrome P450 2B6enzyme
EsketamineCytochrome P450 3A4enzyme
EsketamineCytochrome P450 2C19enzyme
EsketamineCytochrome P450 2C9enzyme
EsketamineGlutamate receptor ionotropic, NMDA 2Btarget
EsketamineElongation factor 2target
EsketamineBrain-derived neurotrophic factortarget
EsketamineBDNF/NT-3 growth factors receptortarget