Isocitrate Dehydrogenase-1 Inhibitors

Name
Isocitrate Dehydrogenase-1 Inhibitors
Accession Number
DBCAT005698
Description

Not Available

Drugs
DrugDrug Description
IvosidenibAn isocitrate dehydrogenase-1 inhibitor used to treat acute myeloid leukemia and cholangiocarcinoma in adults with a susceptible IDH1 mutation.
OlutasidenibAn isocitrate dehydrogenase-1 (IDH1) inhibitor indicated for the treatment of patients with relapsed or refractory acute myeloid leukemia with a susceptible IDH1 mutation as detected by an FDA-approved test.
Drugs & Drug Targets
DrugTargetType
IvosidenibIsocitrate dehydrogenase [NADP] cytoplasmictarget
IvosidenibCytochrome P450 3A4enzyme
IvosidenibCytochrome P450 2B6enzyme
IvosidenibCytochrome P450 2C9enzyme
IvosidenibCytochrome P450 2C8enzyme
IvosidenibSolute carrier family 22 member 8transporter
IvosidenibP-glycoprotein 1transporter
OlutasidenibIsocitrate dehydrogenase [NADP] cytoplasmictarget
OlutasidenibCytochrome P450 3A4enzyme
OlutasidenibCytochrome P450 2C8enzyme
OlutasidenibCytochrome P450 2C9enzyme
OlutasidenibCytochrome P450 1A2enzyme
OlutasidenibCytochrome P450 2C19enzyme
OlutasidenibP-glycoprotein 1transporter
OlutasidenibATP-binding cassette sub-family G member 2transporter
OlutasidenibSolute carrier organic anion transporter family member 1B1transporter
OlutasidenibSolute carrier organic anion transporter family member 1B3transporter
OlutasidenibSolute carrier family 22 member 8transporter
OlutasidenibSolute carrier family 22 member 2transporter
OlutasidenibMultidrug and toxin extrusion protein 1transporter
OlutasidenibMultidrug and toxin extrusion protein 2transporter
OlutasidenibCytochrome P450 2B6enzyme