R-30490

DB09179ExperimentalSmall molecule

R-30490 is an opioid related to carfentanil used as an animal tranquilizer. It was first synthesized by Janssen Pharmaceutica as part of a structure-activity relationship study of fentanly and its... R-30490 was found to be the most selective agonist for the mu opioid receptor out of all the fentanyl analogues tested, but it has never been introduced for medical use in humans, although the closely...

Chemical structure of R-30490
Formula / weight
C24H32N2O2 ยท 380.532 g/mol (avg)
Code names
R 30490

Resolves to

Structure
InChIKeyGARXJOUQUSNOGK-UHFFFAOYSA-NSMILESCCC(=O)N(C1=CC=CC=C1)C1(COC)CCN(CCC2=CC=CC=C2)CC1

Which companies are running trials of R-30490, in which indications and phases, and which of those programs are still active?

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