Tiletamine

DB11549ExperimentalVet approvedSmall molecule

This drug is a dissociative anesthetic agent that falls under the drug category of NMDA receptor antagonists. Tiletamine is chemically similar to another dissociative anesthetic, ketamine. Tiletamine hydrochloride, the salt... Tiletamine hydrochloride, the salt form, exists as odorless white crystals.

Chemical structure of Tiletamine
Mechanism
Curator reviewed
Formula / weight
C12H17NOS · 223.33 g/mol (avg)

Resolves to

Compound
UNII2YFC543249CAS14176-49-9ChEMBLCHEMBL2110703ChEBI94356KEGGD08596
Clinical / RWD
RxNorm1535217
Structure
InChIKeyQAXBVGVYDCAVLV-UHFFFAOYSA-NSMILESCCNC1(CCCCC1=O)C1=CC=CS1

What you can answer from here — as of August 29, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action
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813Drug interactionsStructured to mechanism, not free text
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2Marketed productsAcross 1 country and 1 labeller
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14+ReferencesStructured and connected to the statements they support
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Which companies are running trials of Tiletamine, in which indications and phases, and which of those programs are still active?

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