FAPi-46 GA-68

DB18827InvestigationalSmall molecule

FAPi-46 GA-68: Overview.

Mechanism: Pharmacologically active on Prolyl endopeptidase FAP
Curator reviewed
Formula / weight: C₄₁H₅₄F₂GaN₁₁O₉ · 950.876 g/mol (avg)
Code names: FAPI-46 GA-68

Resolves to

Compound

Structure

[68Ga+3].[H][C@]1(CC(F)(F)CN1C(=O)CNC(=O)C1=CC=NC2=CC=C(C=C12)N(C)CCCN1CCN(CC1)C(=O)CN1CCN(CC([O-])=O)CCN(CC([O-])=O)CCN(CC([O-])=O)CC1)C#N

Targets

What you can answer from here — as of August 31, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

11Clinical trialsPhase, status and sponsor resolved per trial

9+ReferencesStructured and connected to the statements they support

Which drugs share a target with FAPi-46 GA-68, and which of those have an active Phase 3 trial?

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