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Lunresertib

This drug entry is a stub and has not been fully annotated. It is scheduled to be annotated soon.

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Data Packages
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Identification

Generic Name
Lunresertib
DrugBank Accession Number
DB19241
Background

Not Available

Type
Small Molecule
Groups
Investigational
Structure
3D
Similar Structures
Weight
Average: 324.384
Monoisotopic: 324.1586259
Chemical Formula
C18H20N4O2
Synonyms
  • (1S)-2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethyl-1H-Pyrrolo[2,3-b]pyridine-3-carboxamide
External IDs
  • RP-6306
  • RP6306
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Pharmacology

Indication

Not Available

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Contraindications & Blackbox Warnings
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Pharmacodynamics

Not Available

Mechanism of action
Not Available
Absorption

Not Available

Volume of distribution

Not Available

Protein binding

Not Available

Metabolism
Not Available
Route of elimination

Not Available

Half-life

Not Available

Clearance

Not Available

Adverse Effects
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Toxicity

Not Available

Pathways
Not Available
Pharmacogenomic Effects/ADRs
Not Available
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Interactions

Drug Interactions
This information should not be interpreted without the help of a healthcare provider. If you believe you are experiencing an interaction, contact a healthcare provider immediately. The absence of an interaction does not necessarily mean no interactions exist.
Not Available
Food Interactions
Not Available

Categories

Drug Categories
Not Available
Classification
Not classified
Affected organisms
Not Available

Chemical Identifiers

UNII
N95U3A7N57
CAS number
2719793-90-3
InChI Key
ARBRHWRTXPWZGN-UHFFFAOYSA-N
InChI
InChI=1S/C18H20N4O2/c1-8-5-6-13(23)10(3)15(8)22-16(19)14(17(20)24)12-7-9(2)11(4)21-18(12)22/h5-7,23H,19H2,1-4H3,(H2,20,24)
IUPAC Name
SMILES
CC1=C(C)N=C2N(C(N)=C(C(N)=O)C2=C1)C1=C(C)C=CC(O)=C1C

References

General References
Not Available
ChemSpider
115008046
PDBe Ligand
QGI
PDB Entries
8d6e

Clinical Trials

Clinical Trials
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PhaseStatusPurposeConditionsCountStart DateWhy Stopped100+ additional columns
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2RecruitingTreatmentAdvanced Malignant Neoplasm1somestatusstop reasonjust information to hide
2RecruitingTreatmentBreast Cancer1somestatusstop reasonjust information to hide
1Active Not RecruitingTreatmentAdult Solid Tumor1somestatusstop reasonjust information to hide
1Active Not RecruitingTreatmentAdvanced Malignant Neoplasm / Metastatic Cancer / Recurrent Ovarian Cancer / Recurrent Uterine Cancer1somestatusstop reasonjust information to hide
1Active Not RecruitingTreatmentAdvanced Solid Tumors1somestatusstop reasonjust information to hide

Pharmacoeconomics

Manufacturers
Not Available
Packagers
Not Available
Dosage Forms
Not Available
Prices
Not Available
Patents
Not Available

Properties

State
Not Available
Experimental Properties
Not Available
Predicted Properties
PropertyValueSource
Predicted ADMET Features
Not Available

Spectra

Mass Spec (NIST)
Not Available
Spectra
Not Available
Chromatographic Properties
Collision Cross Sections (CCS)
Not Available

Drug created at July 10, 2024 15:06 / Updated at July 11, 2024 07:56