Deltibant

DB20063ExperimentalSmall molecule

Deltibant is a small molecule drug. The usage of the INN stem '-tibant' in the name indicates that Deltibant is a bradykinin receptor antagonist. Deltibant has a monoisotopic molecular weight...

Formula / weight: C₁₂₈H₁₉₄N₄₀O₂₈S₂ · 2805.33 g/mol (avg)
Code names: SB-238592

Resolves to

Compound

UNII6151J4V7VXCAS140661-97-8ChEMBLCHEMBL2103953

Structure

InChIKeyJKUYFMHGTOPVMR-WQVVEKGHSA-NSMILES

CC(C)C[C@H](NC(=O)[C@@H](CC1=CC=CC=C1)NC(=O)[C@H](CS[C@@H]1CC(=O)N(CCCCCCN2C(=O)C[C@H](SC[C@H](NC(=O)[C@H](CC3=CC=CC=C3)NC(=O)CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H]3CCCN3C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](N)CCCNC(N)=N)C(=O)N[C@H](CC3=CC=CC=C3)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(O)=O)C2=O)C1=O)NC(=O)[C@H](CC1=CC=CC=C1)NC(=O)CNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H]1CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](N)CCCNC(N)=N)C(=O)N[C@@H](CCCNC(N)=N)C(O)=O

Targets

P30411BDKRB2

What you can answer from here — as of September 16, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

1+ReferenceStructured and connected to the statements they support

Which drugs share a target with Deltibant, and which of those have an active Phase 3 trial?

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