Palosuran

DB21258ExperimentalSmall molecule

Palosuran is a small molecule drug. The usage of the INN stem '-osuran' in the name indicates that Palosuran is a urotensin receptor antagonist. Palosuran has a monoisotopic molecular weight...

Mechanism: Pharmacologically active on Urotensin-2 receptor
Curator reviewed
Formula / weight: C₂₅H₃₀N₄O₂ · 418.541 g/mol (avg)
Code names: ACT-058362

Resolves to

Compound

UNIIULD9ZKE457CAS540769-28-6ChEMBLCHEMBL567303

Structure

InChIKeyWYJCYXOCHXWTHG-UHFFFAOYSA-NSMILESCC1=NC2=CC=CC=C2C(NC(=O)NCCN2CCC(O)(CC3=CC=CC=C3)CC2)=C1

Targets

Q9UKP6UTS2R

What you can answer from here — as of September 13, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

5+ReferencesStructured and connected to the statements they support

Which drugs share a target with Palosuran, and which of those have an active Phase 3 trial?

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