ATP | investigational, nutraceutical | unknown | target | | Details |
Roxithromycin | approved, investigational, withdrawn | unknown | target | | Details |
Elacridar | investigational | yes | target | inhibitor | Details |
Tesmilifene | investigational | yes | target | inducer | Details |
FM-VP4 | investigational | unknown | target | | Details |
Tariquidar | investigational | yes | target | modulator | Details |
Zosuquidar | investigational | yes | target | inhibitor | Details |
Verapamil | approved | unknown | transporter | substrateinhibitor | Details |
Saquinavir | approved, investigational | unknown | transporter | substrateinhibitorinducer | Details |
Nelfinavir | approved | no | transporter | substrateinhibitorinducer | Details |
Indinavir | approved | unknown | transporter | substrateinhibitorinducer | Details |
Amprenavir | approved, investigational | unknown | transporter | substrateinducer | Details |
Rifampin | approved | unknown | transporter | inducer | Details |
Reserpine | approved, investigational, withdrawn | unknown | transporter | substrateinhibitorinducer | Details |
Nifedipine | approved | unknown | transporter | substrateinducer | Details |
Mifepristone | approved, investigational | unknown | transporter | inhibitorinducer | Details |
Dexamethasone | approved, investigational, vet_approved | unknown | transporter | substrateinhibitorinducer | Details |
Clotrimazole | approved, vet_approved | unknown | transporter | inhibitorinducer | Details |
Carbamazepine | approved, investigational | unknown | transporter | inducer | Details |
Trazodone | approved, investigational | unknown | transporter | inducer | Details |
Nefazodone | approved, withdrawn | unknown | transporter | inhibitorinducer | Details |
Ritonavir | approved, investigational | unknown | transporter | substrateinhibitorinducer | Details |
Digoxin | approved | unknown | transporter | substrateinhibitorinducer | Details |
Liothyronine | approved, vet_approved | unknown | transporter | inducer | Details |
Levothyroxine | approved | unknown | transporter | inducer | Details |
Trimethoprim | approved, vet_approved | unknown | transporter | substrate | Details |
Progesterone | approved, vet_approved | unknown | transporter | substrateinhibitorinducer | Details |
Platelet Activating Factor | experimental | unknown | transporter | substrateinducer | Details |
Cyclosporine | approved, investigational, vet_approved | unknown | transporter | substrateinhibitor | Details |
Cimetidine | approved, investigational | unknown | transporter | substrateinducer | Details |
Aldosterone | experimental, investigational | unknown | transporter | substrateinducer | Details |
Tacrolimus | approved, investigational | unknown | transporter | substrateinhibitorinducer | Details |
Sirolimus | approved, investigational | no | transporter | substrateinhibitorinducer | Details |
Phenobarbital | approved, investigational | unknown | transporter | substrateinducer | Details |
Erythromycin | approved, investigational, vet_approved | no | transporter | substrateinhibitor | Details |
Amiodarone | approved, investigational | unknown | transporter | inhibitorinducer | Details |
St. John's Wort | approved, investigational, nutraceutical | unknown | transporter | inducer | Details |
Vincristine | approved, investigational | unknown | transporter | substrateinhibitorinducer | Details |
Vinblastine | approved | unknown | transporter | substrateinhibitorinducer | Details |
Cholic Acid | approved | unknown | transporter | inducer | Details |
Tamoxifen | approved | unknown | transporter | substrateinhibitorinducer | Details |
Streptozocin | approved, investigational | unknown | transporter | inducer | Details |
Mitoxantrone | approved, investigational | unknown | transporter | substrateinhibitorinducer | Details |
Doxorubicin | approved, investigational | unknown | transporter | substrateinhibitorinducer | Details |
Daunorubicin | approved | unknown | transporter | substrateinhibitorinducer | Details |
Quinidine | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Ketoconazole | approved, investigational | unknown | transporter | inhibitor | Details |
Mibefradil | investigational, withdrawn | unknown | transporter | substrateinhibitor | Details |
Cholesterol | approved, investigational | unknown | transporter | inhibitor | Details |
Mefloquine | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Nicardipine | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Amlodipine | approved | unknown | transporter | substrateinhibitor | Details |
Azelastine | approved | unknown | transporter | inhibitor | Details |
Ranitidine | approved, withdrawn | unknown | transporter | substrateinhibitor | Details |
Etoposide | approved | unknown | transporter | substrateinhibitor | Details |
Methadone | approved | unknown | transporter | inhibitor | Details |
Simvastatin | approved | unknown | transporter | inhibitor | Details |
Lovastatin | approved, investigational | unknown | transporter | inhibitor | Details |
Atorvastatin | approved | no | transporter | substrateinhibitor | Details |
Paclitaxel | approved, vet_approved | unknown | transporter | substrateinhibitor | Details |
Prazosin | approved | unknown | transporter | substrateinhibitormodulator | Details |
Nitrendipine | approved, investigational | unknown | transporter | inhibitor | Details |
Dipyridamole | approved | unknown | transporter | substrateinhibitor | Details |
Diltiazem | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Colchicine | approved | unknown | transporter | substrateinducer | Details |
Clarithromycin | approved | unknown | transporter | substrateinhibitor | Details |
Chlorpromazine | approved, investigational, vet_approved | unknown | transporter | substrateinhibitor | Details |
Dactinomycin | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Troleandomycin | approved | unknown | transporter | inhibitor | Details |
Trifluoperazine | approved, investigational | unknown | transporter | inhibitor | Details |
Terfenadine | approved, withdrawn | unknown | transporter | inhibitor | Details |
Quinine | approved | unknown | transporter | substrateinhibitor | Details |
Itraconazole | approved, investigational | unknown | transporter | inhibitor | Details |
Indomethacin | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Colforsin | experimental, investigational | unknown | transporter | inhibitor | Details |
Fluphenazine | approved | unknown | transporter | inhibitor | Details |
Felodipine | approved, investigational | unknown | transporter | inhibitor | Details |
Carvedilol | approved, investigational | unknown | transporter | inhibitor | Details |
Spironolactone | approved | unknown | transporter | inducer | Details |
Lidocaine | approved, vet_approved | unknown | transporter | inhibitor | Details |
Ciprofloxacin | approved, investigational | unknown | transporter | substrate | Details |
Azithromycin | approved | unknown | transporter | substrateinhibitor | Details |
Acetaminophen | approved | unknown | transporter | substrateinhibitor | Details |
Fluconazole | approved, investigational | unknown | transporter | inhibitor | Details |
Pantoprazole | approved | unknown | transporter | substrateinhibitor | Details |
Omeprazole | approved, investigational, vet_approved | unknown | transporter | substrateinhibitor | Details |
Lansoprazole | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Losartan | approved | unknown | transporter | substrateinhibitor | Details |
Enalapril | approved, vet_approved | unknown | transporter | inhibitor | Details |
Doxazosin | approved | unknown | transporter | inhibitor | Details |
Cilazapril | approved | unknown | transporter | inhibitor | Details |
Captopril | approved | unknown | transporter | inhibitor | Details |
Candesartan cilexetil | approved | unknown | transporter | inhibitor | Details |
Miconazole | approved, investigational, vet_approved | unknown | transporter | inhibitor | Details |
Ergotamine | approved | unknown | transporter | inhibitor | Details |
Ergometrine | approved | unknown | transporter | inhibitor | Details |
Dihydroergotamine | approved, investigational | unknown | transporter | inhibitor | Details |
Bromocriptine | approved, investigational, withdrawn | unknown | transporter | substrateinhibitor | Details |
Loperamide | approved | unknown | transporter | substrate | Details |
Fentanyl | approved, illicit, investigational, vet_approved | unknown | transporter | inhibitor | Details |
Alfentanil | approved, illicit | unknown | transporter | inhibitor | Details |
Nisoldipine | approved | unknown | transporter | inhibitor | Details |
Zimelidine | approved, withdrawn | unknown | transporter | inhibitor | Details |
Tacrine | approved, investigational, withdrawn | unknown | transporter | substrate | Details |
Sumatriptan | approved, investigational | unknown | transporter | substrate | Details |
Selegiline | approved, investigational, vet_approved | unknown | transporter | inhibitor | Details |
Imipramine | approved | unknown | transporter | substrate | Details |
Haloperidol | approved | unknown | transporter | substrateinhibitor | Details |
Fluvoxamine | approved, investigational | unknown | transporter | inhibitor | Details |
Flurazepam | approved, illicit, investigational | unknown | transporter | inhibitor | Details |
Fluoxetine | approved, vet_approved | unknown | transporter | inhibitor | Details |
Doxepin | approved, investigational | unknown | transporter | substrate | Details |
Desipramine | approved, investigational | unknown | transporter | inhibitor | Details |
Clomipramine | approved, investigational, vet_approved | unknown | transporter | inhibitor | Details |
Chlorprothixene | approved, experimental, investigational, withdrawn | unknown | transporter | inhibitor | Details |
Buspirone | approved, investigational | unknown | transporter | inhibitor | Details |
Pimozide | approved | unknown | transporter | inhibitor | Details |
Morphine | approved, investigational | no | transporter | substrate | Details |
Ivermectin | approved, investigational, vet_approved | unknown | transporter | substrateinhibitorinducer | Details |
Hydrocortisone | approved, vet_approved | unknown | transporter | substrateinducer | Details |
Astemizole | approved, withdrawn | unknown | transporter | inhibitor | Details |
Triflupromazine | approved, vet_approved | unknown | transporter | inhibitor | Details |
Protriptyline | approved | unknown | transporter | inhibitor | Details |
Promethazine | approved, investigational | unknown | transporter | inhibitor | Details |
Bepridil | approved, withdrawn | unknown | transporter | inhibitor | Details |
Loratadine | approved, investigational | no | transporter | substrateinhibitor | Details |
Desloratadine | approved, investigational | unknown | transporter | inhibitor | Details |
Venlafaxine | approved | unknown | transporter | substrateinhibitor | Details |
Sertraline | approved | unknown | transporter | inhibitor | Details |
Reboxetine | approved, experimental | unknown | transporter | inhibitor | Details |
Paroxetine | approved, investigational | unknown | transporter | inhibitor | Details |
Citalopram | approved | unknown | transporter | substrateinhibitor | Details |
Estramustine | approved, investigational | unknown | transporter | inhibitor | Details |
Taurocholic acid | approved, experimental | unknown | transporter | substrateinhibitor | Details |
Flupentixol | approved, investigational, withdrawn | unknown | transporter | inhibitor | Details |
Megestrol acetate | approved, investigational, vet_approved | unknown | transporter | inhibitor | Details |
Staurosporine | experimental | unknown | transporter | inhibitor | Details |
Quinacrine | investigational | unknown | transporter | inhibitor | Details |
Genistein | investigational | unknown | transporter | inhibitor | Details |
Quercetin | experimental, investigational | unknown | transporter | inhibitor | Details |
Levofloxacin | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Naringenin | experimental | unknown | transporter | downregulator | Details |
Glyburide | approved | unknown | transporter | inhibitor | Details |
Fexofenadine | approved, investigational | unknown | transporter | substrate | Details |
Trimipramine | approved | unknown | transporter | substrate | Details |
Propranolol | approved, investigational | unknown | transporter | substrate | Details |
Prednisone | approved, vet_approved | unknown | transporter | substrateinducer | Details |
Amsacrine | approved, investigational | unknown | transporter | inhibitor | Details |
Gramicidin D | approved | unknown | transporter | substrateinhibitor | Details |
Benzocaine | approved, investigational | unknown | transporter | inhibitor | Details |
Lopinavir | approved | unknown | transporter | inhibitorinducer | Details |
Caspofungin | approved | unknown | transporter | inhibitor | Details |
Pravastatin | approved | no | transporter | substrate | Details |
Imatinib | approved | no | transporter | substrateinhibitor | Details |
Sorafenib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Sunitinib | approved, investigational | unknown | transporter | inhibitor | Details |
Terazosin | approved | unknown | transporter | inhibitor | Details |
Dronabinol | approved, illicit | unknown | transporter | inhibitor | Details |
Buprenorphine | approved, illicit, investigational, vet_approved | unknown | transporter | inhibitor | Details |
Telmisartan | approved, investigational | unknown | transporter | inhibitor | Details |
Dasatinib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Gefitinib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Nilotinib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Estrone | approved | unknown | transporter | substrateinducer | Details |
Lapatinib | approved, investigational | unknown | transporter | inhibitor | Details |
Posaconazole | approved, investigational, vet_approved | unknown | transporter | substrateinhibitor | Details |
Grepafloxacin | approved, investigational, withdrawn | unknown | transporter | substrateinhibitor | Details |
Diazepam | approved, illicit, investigational, vet_approved | unknown | transporter | substrate | Details |
Digitoxin | approved, investigational | unknown | transporter | substrate | Details |
Sparfloxacin | approved, investigational, withdrawn | unknown | transporter | substrate | Details |
Methylprednisolone | approved, vet_approved | unknown | transporter | substrateinducer | Details |
Quetiapine | approved | unknown | transporter | substrate | Details |
Olanzapine | approved, investigational | no | transporter | substrate | Details |
Clozapine | approved | unknown | transporter | substrate | Details |
Naloxone | approved, vet_approved | unknown | transporter | substrate | Details |
Camptothecin | experimental | unknown | transporter | substrate | Details |
Prednisolone | approved, vet_approved | unknown | transporter | substrate | Details |
Acebutolol | approved, investigational | unknown | transporter | substrate | Details |
Ibuprofen | approved | unknown | transporter | substrate | Details |
Acetylsalicylic acid | approved, vet_approved | unknown | transporter | substrateinducermodulator | Details |
Domperidone | approved, investigational, vet_approved | unknown | transporter | substrate | Details |
Betamethasone | approved, vet_approved | unknown | transporter | substrate | Details |
Toremifene | approved, investigational | unknown | transporter | substrate | Details |
Diethylstilbestrol | approved, investigational, withdrawn | unknown | transporter | substrate | Details |
Clomifene | approved, investigational | unknown | transporter | substrate | Details |
Estradiol | approved, investigational, vet_approved | unknown | transporter | substratedownregulatorregulator | Details |
Docetaxel | approved, investigational | unknown | transporter | substrate | Details |
Methotrexate | approved | unknown | transporter | substrate | Details |
Timolol | approved | unknown | transporter | substrate | Details |
Nadolol | approved | unknown | transporter | substrate | Details |
Alitretinoin | approved, investigational | unknown | transporter | substrate | Details |
Vecuronium | approved, investigational | unknown | transporter | substrate | Details |
Debrisoquine | approved, investigational | unknown | transporter | substrate | Details |
Gemcitabine | approved | no | transporter | substrate | Details |
Topotecan | approved, investigational | unknown | transporter | substrate | Details |
Stanolone | illicit, investigational | unknown | transporter | substrate | Details |
Epinastine | approved, investigational | unknown | transporter | substrate | Details |
Norethisterone | approved | unknown | transporter | inhibitor | Details |
Estriol | approved, investigational, vet_approved | unknown | transporter | substrateinducer | Details |
Sphingosine | experimental | unknown | transporter | substrate | Details |
Cerivastatin | approved, withdrawn | unknown | transporter | substrate | Details |
Conjugated estrogens | approved | unknown | transporter | substrate | Details |
Levetiracetam | approved | unknown | transporter | substrate | Details |
Phenytoin | approved, vet_approved | unknown | transporter | substrate | Details |
Nizatidine | approved | unknown | transporter | substrate | Details |
Erlotinib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Lamotrigine | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Sitagliptin | approved, investigational | unknown | transporter | substrate | Details |
Atazanavir | approved, investigational | unknown | transporter | substrateinhibitorinducer | Details |
Arsenic trioxide | approved, investigational | unknown | transporter | inhibitor | Details |
Cabazitaxel | approved | unknown | transporter | substrateinhibitor | Details |
Liotrix | approved | unknown | transporter | inducer | Details |
Temsirolimus | approved | unknown | transporter | substrateinhibitor | Details |
Ketazolam | approved | unknown | transporter | substrate | Details |
Voacamine | experimental | unknown | target | inhibitor | Details |
Ethinylestradiol | approved | unknown | transporter | substrate | Details |
Propafenone | approved | unknown | transporter | inhibitor | Details |
Eletriptan | approved, investigational | unknown | transporter | substrate | Details |
Dronedarone | approved | no | transporter | inhibitor | Details |
Romidepsin | approved, investigational | unknown | transporter | substrate | Details |
Silodosin | approved | unknown | transporter | substrate | Details |
Etravirine | approved | unknown | transporter | inhibitor | Details |
Rivaroxaban | approved | unknown | transporter | substrate | Details |
Dabigatran etexilate | approved | unknown | transporter | substrate | Details |
Ezetimibe | approved | unknown | transporter | substrate | Details |
Fesoterodine | approved | unknown | transporter | substrate | Details |
Tolvaptan | approved | no | transporter | substrateinhibitor | Details |
Pitavastatin | approved | unknown | transporter | substrate | Details |
Pazopanib | approved | unknown | transporter | substrate | Details |
Rilpivirine | approved | unknown | transporter | inhibitor | Details |
Boceprevir | approved, withdrawn | unknown | transporter | inhibitor | Details |
Telaprevir | approved, withdrawn | unknown | transporter | substrateinhibitor | Details |
Fidaxomicin | approved | no | transporter | substrate | Details |
Indacaterol | approved | unknown | transporter | substrate | Details |
Clobazam | approved, illicit | no | transporter | substrate | Details |
Linagliptin | approved | unknown | transporter | substrate | Details |
Lomitapide | approved, investigational | no | transporter | inhibitor | Details |
Ticagrelor | approved | unknown | transporter | substrateinhibitor | Details |
Crizotinib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Apixaban | approved | unknown | transporter | substrate | Details |
Axitinib | approved, investigational | no | transporter | substrateinhibitor | Details |
Vismodegib | approved, investigational | unknown | transporter | substrate | Details |
Carfilzomib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Mirabegron | approved | unknown | transporter | substrateinhibitor | Details |
Regorafenib | approved | unknown | transporter | substrateinhibitor | Details |
Enzalutamide | approved | no | transporter | inhibitor | Details |
Ivacaftor | approved | no | transporter | inhibitor | Details |
Bosutinib | approved | no | transporter | substrate | Details |
Ponatinib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Fluticasone furoate | approved | no | transporter | substrateinducer | Details |
Canagliflozin | approved | unknown | transporter | substrateinhibitor | Details |
Pomalidomide | approved | unknown | transporter | substrate | Details |
Lenalidomide | approved | no | transporter | substrate | Details |
Dabrafenib | approved, investigational | no | transporter | substrate | Details |
Trastuzumab emtansine | approved, investigational | unknown | transporter | substrate | Details |
Zidovudine | approved | unknown | transporter | substrate | Details |
Clopidogrel | approved | no | transporter | substrate | Details |
Afatinib | approved | unknown | transporter | substrateinhibitor | Details |
Irinotecan | approved, investigational | unknown | transporter | substrate | Details |
Lamivudine | approved, investigational | unknown | transporter | substrate | Details |
Mycophenolate mofetil | approved, investigational | unknown | transporter | substrate | Details |
Levomilnacipran | approved, investigational | unknown | transporter | substrate | Details |
Simeprevir | approved | unknown | transporter | substrateinhibitor | Details |
Sofosbuvir | approved | no | transporter | substrate | Details |
Dapagliflozin | approved | unknown | transporter | substrate | Details |
Umeclidinium | approved | no | transporter | substrate | Details |
Edoxaban | approved | no | transporter | substrate | Details |
Ceritinib | approved | no | transporter | substrate | Details |
Lenvatinib | approved, investigational | no | transporter | substrateinhibitor | Details |
Nintedanib | approved | no | transporter | substrateinhibitor | Details |
Idelalisib | approved | no | transporter | substrateinhibitor | Details |
Cobicistat | approved | unknown | transporter | inhibitor | Details |
Rolapitant | approved, investigational | no | transporter | inhibitor | Details |
Daclatasvir | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Isavuconazonium | approved, investigational | no | transporter | inhibitor | Details |
Panobinostat | approved, investigational | no | transporter | substrate | Details |
Osimertinib | approved | no | transporter | substrate | Details |
Selexipag | approved | no | transporter | substrate | Details |
Ambrisentan | approved, investigational | unknown | transporter | substrate | Details |
Ombitasvir | approved, investigational | no | transporter | substrate | Details |
Elbasvir | approved | no | transporter | substrateinhibitor | Details |
Grazoprevir | approved | no | transporter | substrate | Details |
Technetium Tc-99m sestamibi | approved, investigational | no | transporter | substrate | Details |
Venetoclax | approved, investigational | no | transporter | substrateinhibitor | Details |
Belinostat | approved, investigational | unknown | transporter | substrate | Details |
Velpatasvir | approved, investigational | no | transporter | substrateinhibitor | Details |
Ledipasvir | approved | no | transporter | substratetransporter | Details |
Lobeglitazone | experimental | no | transporter | | Details |
Miltefosine | approved, investigational | unknown | target | | Details |
Lumacaftor | approved | no | transporter | inhibitorinducer | Details |
Neratinib | approved, investigational | unknown | transporter | inhibitor | Details |
Voxilaprevir | approved, investigational | no | transporter | substrateinhibitor | Details |
Enasidenib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Inotuzumab ozogamicin | approved, investigational | unknown | transporter | substrate | Details |
Pibrentasvir | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Glecaprevir | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Copanlisib | approved, investigational | unknown | transporter | substrate | Details |
Abemaciclib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Betrixaban | approved, investigational | no | transporter | substrate | Details |
Candesartan | experimental | unknown | transporter | inhibitor | Details |
Letermovir | approved, investigational | no | transporter | substrateinhibitor | Details |
Rucaparib | approved, investigational | no | transporter | substrateinhibitor | Details |
Ubidecarenone | approved, investigational, nutraceutical | no | transporter | substrate | Details |
Ertugliflozin | approved, investigational | no | transporter | substrate | Details |
Testosterone cypionate | approved | unknown | transporter | inhibitor | Details |
Testosterone enanthate | approved | unknown | transporter | inhibitor | Details |
Testosterone undecanoate | approved, investigational | unknown | transporter | inhibitor | Details |
Technetium Tc-99m tetrofosmin | approved | no | carrier | binder | Details |
Stanolone acetate | experimental | unknown | transporter | substrate | Details |
Estradiol acetate | approved, investigational, vet_approved | unknown | transporter | substrate | Details |
Estradiol benzoate | approved, investigational, vet_approved | unknown | transporter | substrate | Details |
Estradiol cypionate | approved, investigational, vet_approved | unknown | transporter | substrate | Details |
Estradiol dienanthate | approved, investigational, vet_approved | unknown | transporter | substrate | Details |
Estradiol valerate | approved, investigational, vet_approved | unknown | transporter | substrate | Details |
Testosterone propionate | approved, investigational, vet_approved, withdrawn | no | transporter | substrate | Details |
Apalutamide | approved, investigational | unknown | transporter | inducer | Details |
Isavuconazole | approved, investigational | unknown | transporter | inhibitor | Details |
Tocopherol | approved, investigational | no | transporter | transporter | Details |
alpha-Tocopherol acetate | approved | no | transporter | substrate | Details |
Somatostatin | approved, investigational | unknown | transporter | substrate | Details |
Tocofersolan | approved | yes | target | antagonist | Details |
Vinflunine | approved, investigational | no | transporter | substrate | Details |
Curcumin | approved, investigational | unknown | transporter | inhibitor | Details |
Avatrombopag | approved, investigational | no | transporter | substrate | Details |
Paritaprevir | approved, investigational | unknown | transporter | substrate | Details |
Dasabuvir | approved | unknown | transporter | substrate | Details |
Fentanyl | approved, illicit, investigational, vet_approved | unknown | target | | Details |
Concanamycin A | experimental | yes | target | inhibitor | Details |
Hycanthone | experimental | yes | target | inhibitor | Details |
Dexverapamil | experimental | yes | target | inhibitor | Details |
Emopamil | experimental | yes | target | inhibitor | Details |
Lomerizine | experimental | yes | target | inhibitor | Details |
Tetrandrine | experimental | unknown | target | inhibitor | Details |
Dofequidar | experimental, investigational | unknown | target | inhibitor | Details |
Dexniguldipine | experimental | unknown | target | inhibitor | Details |
ONT-093 | investigational | yes | target | inhibitor | Details |
HM-30181 | experimental | yes | target | inhibitor | Details |
Desmethylsertraline | experimental | unknown | target | inhibitor | Details |
Reversin 121 | experimental | yes | target | inhibitor | Details |
Loxicodegol | investigational | unknown | transporter | | Details |
Hydrocortisone aceponate | experimental, vet_approved | unknown | transporter | | Details |
Hydrocortisone acetate | approved, vet_approved | unknown | transporter | | Details |
Hydrocortisone butyrate | approved, vet_approved | unknown | transporter | | Details |
Hydrocortisone cypionate | approved, investigational, vet_approved | unknown | transporter | | Details |
Hydrocortisone phosphate | approved, vet_approved | unknown | transporter | | Details |
Hydrocortisone probutate | approved, vet_approved | unknown | transporter | | Details |
Hydrocortisone valerate | approved, vet_approved | unknown | transporter | | Details |
Ivosidenib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Elagolix | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Fluticasone | approved, experimental | no | carrier | substrate | Details |
Chloroquine | approved, investigational, vet_approved | unknown | transporter | substrateinhibitor | Details |
Amodiaquine | approved, investigational | unknown | transporter | inhibitor | Details |
Primaquine | approved | unknown | transporter | inhibitor | Details |
Hydroxychloroquine | approved | unknown | transporter | inhibitor | Details |
Paliperidone | approved | unknown | transporter | substrateinhibitor | Details |
Dovitinib | investigational | unknown | transporter | inhibitor | Details |
Lusutrombopag | approved, investigational | unknown | transporter | substrate | Details |
Curcumin sulfate | experimental | unknown | transporter | | Details |
Estriol tripropionate | experimental | unknown | transporter | | Details |
Duvelisib | approved, investigational | no | transporter | substrate | Details |
Dexibuprofen | approved, investigational | unknown | transporter | | Details |
Talazoparib | approved, investigational | unknown | transporter | substrate | Details |
Omadacycline | approved, investigational | unknown | transporter | substrate | Details |
Grapiprant | investigational, vet_approved | no | transporter | substrate | Details |
Sarecycline | approved, investigational | unknown | transporter | inhibitor | Details |
Rifamycin | approved, investigational | no | transporter | substrateinhibitor | Details |
Dacomitinib | approved, investigational | no | transporter | substrateinhibitor | Details |
Revefenacin | approved, investigational | no | transporter | substrate | Details |
Gilteritinib | approved, investigational | no | transporter | substrate | Details |
Tenofovir | experimental, investigational | no | transporter | substrate | Details |
Tenofovir disoproxil | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Tenofovir alafenamide | approved | unknown | transporter | substrate | Details |
Darunavir | approved | unknown | transporter | substrateinhibitorinducer | Details |
Sildenafil | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Vardenafil | approved | unknown | transporter | substrateinhibitor | Details |
Oxcarbazepine | approved | unknown | transporter | substrate | Details |
Cabergoline | approved | no | transporter | substrate | Details |
Prucalopride | approved | no | transporter | substrate | Details |
Risperidone | approved, investigational | unknown | transporter | substrate | Details |
Atovaquone | approved | no | transporter | inhibitor | Details |
Naproxen | approved, vet_approved | no | transporter | inhibitor | Details |
Rifabutin | approved, investigational | unknown | transporter | inducer | Details |
Piperine | investigational | unknown | transporter | inhibitor | Details |
Glasdegib | approved, investigational | no | transporter | substrateinhibitor | Details |
Olaparib | approved | no | transporter | substrateinhibitor | Details |
Ranolazine | approved, investigational | no | transporter | substrateinhibitor | Details |
Amitriptyline | approved | unknown | transporter | substrate | Details |
Cetirizine | approved | no | transporter | substrateinhibitor | Details |
Palbociclib | approved, investigational | no | transporter | substrateinhibitor | Details |
Tegaserod | approved, investigational, withdrawn | unknown | transporter | substrate | Details |
Fluticasone | approved, experimental | unknown | transporter | substrate | Details |
Erdafitinib | approved, investigational | no | transporter | substrateinhibitor | Details |
Esomeprazole | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Duloxetine | approved | unknown | transporter | inhibitor | Details |
Raloxifene | approved, investigational | unknown | transporter | substrate | Details |
Alpelisib | approved, investigational | unknown | transporter | inhibitor | Details |
Tezacaftor | approved, investigational | no | transporter | substrateinhibitor | Details |
Olopatadine | approved | no | transporter | substrate | Details |
Nitrofurantoin | approved, vet_approved | unknown | transporter | substrate | Details |
Levothyroxine | approved | no | enzyme | inducer | Details |
Beclomethasone dipropionate | approved, investigational | unknown | transporter | substrateinducer | Details |
Bisoprolol | approved | unknown | transporter | substrateinhibitor | Details |
Metronidazole | approved | unknown | transporter | inhibitor | Details |
Celecoxib | approved, investigational | unknown | transporter | substrate | Details |
Entrectinib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Fedratinib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Lefamulin | approved, investigational | unknown | transporter | substrate | Details |
Budesonide | approved | no | transporter | substrate | Details |
Istradefylline | approved, investigational | unknown | transporter | inhibitor | Details |
Metoclopramide | approved, investigational | unknown | transporter | substrate | Details |
Escitalopram | approved | unknown | transporter | substrate | Details |
Medroxyprogesterone acetate | approved, investigational | unknown | target | inhibitor | Details |
Anastrozole | approved, investigational | unknown | transporter | substrate | Details |
Flecainide | approved, withdrawn | unknown | transporter | substrate | Details |
Acenocoumarol | approved, investigational | unknown | transporter | substrate | Details |
Apremilast | approved, investigational | unknown | transporter | substrate | Details |
Lasmiditan | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Asunaprevir | approved, investigational, withdrawn | unknown | transporter | substrateinhibitor | Details |
Elexacaftor | approved, investigational | no | transporter | substrateinhibitor | Details |
Prednisolone acetate | approved, vet_approved | unknown | transporter | substrate | Details |
Zanubrutinib | approved, investigational | no | transporter | substrate | Details |
Topiramate | approved | unknown | transporter | substrate | Details |
Levamlodipine | approved, investigational | unknown | transporter | substrate | Details |
Trastuzumab deruxtecan | approved, investigational | no | transporter | substrate | Details |
Enfortumab vedotin | approved, investigational | unknown | transporter | substrate | Details |
Lemborexant | approved, investigational | unknown | transporter | substrate | Details |
Darolutamide | approved, investigational | unknown | transporter | substrate | Details |
Upadacitinib | approved, investigational | no | transporter | substrateinhibitor | Details |
Ubrogepant | approved, investigational | unknown | transporter | substrate | Details |
Avapritinib | approved, investigational | unknown | transporter | inhibitormodulator | Details |
Azathioprine | approved | unknown | transporter | substrate | Details |
Hydroxyzine | approved | unknown | transporter | substrate | Details |
Polyethylene glycol 400 | approved | unknown | transporter | inhibitor | Details |
Tazemetostat | approved, investigational | unknown | transporter | substrate | Details |
Letrozole | approved, investigational | unknown | transporter | substrate | Details |
Ziprasidone | approved | unknown | transporter | | Details |
Clindamycin | approved, vet_approved | unknown | transporter | substrate | Details |
Polyethylene glycol | approved, vet_approved | no | transporter | inhibitor | Details |
Norgestimate | approved, investigational | unknown | transporter | inhibitor | Details |
Talinolol | investigational | unknown | transporter | substrate | Details |
Elacridar | investigational | unknown | transporter | inhibitor | Details |
Tipranavir | approved, investigational | unknown | transporter | substrateinhibitorinducer | Details |
Valspodar | investigational | unknown | transporter | inhibitor | Details |
Albendazole | approved, vet_approved | no | transporter | substrate | Details |
Cobimetinib | approved, investigational | no | transporter | substrate | Details |
Odanacatib | investigational | unknown | transporter | substrate | Details |
Voacamine | experimental | no | transporter | inhibitor | Details |
Dolutegravir | approved | no | transporter | substrate | Details |
Diclofenac | approved, vet_approved | unknown | transporter | inducer | Details |
Baricitinib | approved, investigational | unknown | transporter | substrate | Details |
Alectinib | approved, investigational | unknown | transporter | inhibitor | Details |
Larotrectinib | approved, investigational | no | transporter | substrate | Details |
Fluticasone propionate | approved | unknown | transporter | substrate | Details |
Monensin | experimental, vet_approved | unknown | transporter | substrate | Details |
Rhodamine 6G | experimental | unknown | transporter | substrate | Details |
Niguldipine | experimental | unknown | transporter | inhibitor | Details |
Biricodar | investigational | unknown | transporter | inhibitor | Details |
Tariquidar | investigational | unknown | transporter | inhibitor | Details |
Laniquidar | investigational | unknown | transporter | inhibitor | Details |
Gallopamil | investigational | unknown | transporter | inhibitor | Details |
Annamycin | investigational | unknown | transporter | | Details |
Nortriptyline | approved | unknown | transporter | substrate | Details |
Meperidine | approved | unknown | transporter | substrate | Details |
Pentazocine | approved, vet_approved | unknown | transporter | substrate | Details |
Propofol | approved, investigational, vet_approved | unknown | transporter | inducer | Details |
Everolimus | approved | unknown | transporter | substrateinhibitor | Details |
Ceftriaxone | approved | unknown | transporter | inhibitor | Details |
Conivaptan | approved, investigational | unknown | transporter | inhibitor | Details |
Salinomycin | vet_approved | unknown | transporter | inhibitor | Details |
Zonisamide | approved, investigational | unknown | transporter | inhibitor | Details |
Valinomycin | experimental | unknown | transporter | substrateinhibitor | Details |
Flibanserin | approved, investigational | unknown | transporter | inhibitor | Details |
Eliglustat | approved, investigational | no | transporter | substrateinhibitor | Details |
Bicalutamide | approved | unknown | transporter | inhibitor | Details |
Mitotane | approved | unknown | transporter | inhibitor | Details |
Lonafarnib | approved, investigational | no | transporter | substrateinhibitor | Details |
Tipifarnib | investigational | unknown | transporter | inhibitor | Details |
Netupitant | approved, investigational | unknown | transporter | inhibitor | Details |
Suvorexant | approved, investigational | unknown | transporter | | Details |
Vorapaxar | approved | unknown | transporter | | Details |
Vandetanib | approved | unknown | transporter | inhibitor | Details |
Concanamycin A | experimental | unknown | transporter | inhibitor | Details |
Hycanthone | experimental | unknown | transporter | inhibitor | Details |
Vemurafenib | approved | unknown | transporter | substrateinhibitor | Details |
Dexverapamil | experimental | unknown | transporter | inhibitor | Details |
Emopamil | experimental | unknown | transporter | inhibitor | Details |
Lomerizine | experimental | unknown | transporter | inhibitor | Details |
Tetrandrine | experimental | unknown | transporter | inhibitor | Details |
ONT-093 | investigational | unknown | transporter | inhibitor | Details |
Dofequidar | experimental, investigational | unknown | transporter | inhibitor | Details |
Medroxyprogesterone acetate | approved, investigational | unknown | transporter | inhibitor | Details |
Rimegepant | approved, investigational | unknown | transporter | substrate | Details |
Favipiravir | approved, investigational | unknown | transporter | inhibitor | Details |
Medrysone | approved | unknown | transporter | substrate | Details |
Methylene blue | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Ozanimod | approved, investigational | unknown | transporter | substrate | Details |
Fingolimod | approved, investigational | no | transporter | inhibitor | Details |
Chloramphenicol succinate | approved | unknown | transporter | substrate | Details |
Selumetinib | approved, investigational | unknown | transporter | substrate | Details |
Prednisolone phosphate | approved, vet_approved | unknown | transporter | substrateinducer | Details |
Tucatinib | approved, investigational | unknown | transporter | substrate | Details |
Pemigatinib | approved, investigational | no | transporter | substrateinhibitor | Details |
Zolmitriptan | approved, investigational | no | transporter | | Details |
Remdesivir | approved, investigational | unknown | transporter | substrate | Details |
Capmatinib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Ixabepilone | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Selpercatinib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Ripretinib | approved | unknown | transporter | substrateinhibitor | Details |
Clofazimine | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Empagliflozin | approved | unknown | transporter | substrate | Details |
Cethromycin | investigational | unknown | transporter | substrateinhibitor | Details |
Galantamine | approved | no | transporter | inhibitor | Details |
Aliskiren | approved, investigational | no | transporter | substrate | Details |
Artesunate | approved, investigational | unknown | transporter | substrate | Details |
Bortezomib | approved, investigational | no | transporter | substrate | Details |
Betamethasone phosphate | approved, vet_approved | unknown | transporter | substrateinducer | Details |
Lurbinectedin | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Dexamethasone acetate | approved, investigational, vet_approved | unknown | transporter | substrateinhibitorinducer | Details |
Octreotide | approved, investigational | unknown | transporter | substrate | Details |
Fostemsavir | approved, investigational | unknown | transporter | substrate | Details |
Belantamab mafodotin | approved | unknown | transporter | substrate | Details |
Risdiplam | approved, investigational | unknown | transporter | substrate | Details |
Pralsetinib | approved, investigational | no | transporter | substrateinhibitor | Details |
Filgotinib | approved, investigational | unknown | transporter | substrate | Details |
Berotralstat | approved | no | transporter | substrateinhibitor | Details |
Relugolix | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Vibegron | approved, investigational | no | transporter | substrate | Details |
Cortisone acetate | approved, investigational | unknown | transporter | substrateinducer | Details |
Opicapone | approved, investigational | no | transporter | substrate | Details |
Vericiguat | approved, investigational | unknown | transporter | substrate | Details |
Cabotegravir | approved, investigational | unknown | transporter | substrate | Details |
Voclosporin | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Tepotinib | approved, investigational | no | transporter | substrateinhibitor | Details |
Somatotropin | approved, investigational | unknown | transporter | substrate | Details |
Alfuzosin | approved, investigational | unknown | transporter | substrate | Details |
Trilaciclib | approved, investigational | unknown | transporter | substrate | Details |
Umbralisib | approved, investigational, withdrawn | unknown | transporter | inhibitor | Details |
Sulpiride | approved, investigational | unknown | transporter | substrate | Details |
Temozolomide | approved, investigational | no | transporter | substrate | Details |
Avanafil | approved | unknown | transporter | substrate | Details |
Tivozanib | approved, investigational | unknown | transporter | substrate | Details |
Daptomycin | approved, investigational | no | transporter | substrate | Details |
Amisulpride | approved, investigational | no | transporter | substrate | Details |
Diosmin | approved, investigational | unknown | transporter | inhibitor | Details |
Vildagliptin | approved, investigational | no | transporter | substrate | Details |
Azilsartan medoxomil | approved, investigational | no | transporter | inhibitor | Details |
Sapropterin | approved, investigational | unknown | transporter | inhibitor | Details |
Levoketoconazole | approved, investigational | no | transporter | inhibitor | Details |
Loncastuximab tesirine | approved, investigational | unknown | transporter | substrate | Details |
Sotorasib | approved, investigational | unknown | transporter | inhibitor | Details |
Infigratinib | approved, investigational | no | transporter | substrateinhibitor | Details |
Ibrexafungerp | approved, investigational | unknown | transporter | substratetransporter | Details |
Belumosudil | approved, investigational | no | transporter | substrateinhibitor | Details |
Odevixibat | approved, investigational | unknown | transporter | substrate | Details |
Belzutifan | approved, investigational | no | transporter | substrate | Details |
Lonapegsomatropin | approved, investigational | unknown | transporter | substrate | Details |
Mobocertinib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Tisotumab vedotin | approved | no | transporter | substrate | Details |
Atogepant | approved, investigational | no | transporter | substrate | Details |
Riociguat | approved | no | transporter | substrate | Details |
Avacopan | approved, investigational | no | transporter | substrate | Details |
Asciminib | approved, investigational | no | transporter | substrateinhibitor | Details |
Maribavir | approved, investigational | no | transporter | inhibitor | Details |
Nirmatrelvir | approved, investigational | no | transporter | substrateinhibitor | Details |
Sotagliflozin | approved, investigational | no | transporter | inhibitor | Details |
Abrocitinib | approved, investigational | unknown | transporter | inhibitor | Details |
Mitapivat | approved, investigational | no | transporter | substrateinhibitor | Details |
Cannabidiol | approved, investigational | no | transporter | inhibitor | Details |
Cannabinol | experimental, investigational | unknown | transporter | inhibitor | Details |
Medical Cannabis | experimental, investigational | unknown | transporter | inhibitor | Details |
Pacritinib | approved, investigational | no | transporter | inhibitor | Details |
Cariprazine | approved, investigational | unknown | transporter | inhibitor | Details |
Azvudine | investigational | unknown | target | activatorregulator | Details |
SAR-405838 | investigational | no | transporter | substrate | Details |
Verapamil | approved | unknown | target | inhibitorblocker | Details |
Stiripentol | approved | unknown | transporter | inhibitor | Details |
Pirfenidone | approved, investigational | unknown | transporter | inhibitor | Details |
Baloxavir marboxil | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Lenacapavir | approved, investigational | no | transporter | substrate | Details |
Deucravacitinib | approved, investigational | unknown | transporter | substrate | Details |
Telotristat ethyl | approved, investigational | no | transporter | substrateinhibitor | Details |
Futibatinib | approved, investigational | no | transporter | substrateinhibitor | Details |
Vonoprazan | approved, investigational | unknown | transporter | inhibitor | Details |
Niraparib | approved, investigational | no | transporter | substrate | Details |
Mirvetuximab soravtansine | approved, investigational | no | transporter | substrate | Details |
Olutasidenib | approved, investigational | no | transporter | inhibitor | Details |
Polatuzumab vedotin | approved, investigational | no | transporter | substrate | Details |
Adagrasib | approved, investigational | unknown | transporter | inhibitor | Details |
Bexagliflozin | approved, investigational | unknown | transporter | substrate | Details |
Pirtobrutinib | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Elacestrant | approved, investigational | unknown | transporter | inhibitor | Details |
Midazolam | approved, illicit | no | transporter | substrate | Details |
Sparsentan | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Zavegepant | approved, investigational | unknown | transporter | substrate | Details |
Leniolisib | approved, investigational | no | transporter | substrate | Details |
Aripiprazole | approved, investigational | unknown | transporter | inhibitor | Details |
Vilanterol | approved | no | transporter | substrate | Details |
Quizartinib | approved, investigational | no | transporter | substrateinhibitor | Details |
Momelotinib | approved, investigational | unknown | transporter | substrate | Details |
Encorafenib | approved, investigational | no | transporter | substrateinhibitor | Details |
Gefapixant | approved, investigational | no | transporter | substrate | Details |
Binimetinib | approved, investigational | no | transporter | substrate | Details |
Repotrectinib | approved, investigational | no | transporter | substrateinhibitor | Details |
Nirogacestat | approved, investigational | no | transporter | substrateinhibitor | Details |
Aprocitentan | approved, investigational | no | transporter | substrate | Details |
Danicopan | approved, investigational | no | transporter | inhibitor | Details |
Mavorixafor | approved, investigational | unknown | transporter | substrateinhibitor | Details |
Cladribine | approved, investigational | unknown | transporter | substrate | Details |
Deuruxolitinib | investigational | unknown | transporter | substrate | Details |
Seladelpar | approved, investigational | unknown | transporter | substrate | Details |
Biricodar | investigational | yes | target | modulator | Details |
Ixazomib | approved, investigational | unknown | transporter | substrate | Details |
L-Acetylleucine | approved, investigational | no | transporter | inhibitor | Details |
Benzgalantamine | approved | no | transporter | inhibitor | Details |