Fludiazepam | experimental, illicit | yes | target | potentiator | Details |
Ethanol | approved | unknown | target | | Details |
Ocinaplon | investigational | yes | target | modulator | Details |
ORG-25435 | investigational | yes | target | modulator | Details |
AZD-3043 | investigational | yes | target | modulator | Details |
EVT 201 | investigational | yes | target | modulator | Details |
Pagoclone | investigational | yes | target | modulator | Details |
Zuranolone | approved, experimental | yes | target | modulator | Details |
Clomethiazole | investigational | yes | target | modulator | Details |
Arbaclofen Placarbil | investigational | yes | target | agonist | Details |
Remimazolam | approved, investigational | yes | target | agonist | Details |
Bentazepam | experimental | yes | target | modulator | Details |
Stiripentol | approved | yes | target | modulator | Details |
Zolpidem | approved | yes | target | allosteric modulator | Details |
Flumazenil | approved | yes | target | allosteric modulator | Details |
Mebutamate | approved | yes | target | modulator | Details |
Metharbital | withdrawn | yes | target | modulator | Details |
Etomidate | approved | yes | target | modulator | Details |
Thiamylal | approved, vet_approved | yes | target | modulator | Details |
Clobazam | approved, illicit | yes | target | modulator | Details |
Talbutal | approved, illicit | yes | target | modulator | Details |
Brexanolone | approved, investigational | yes | target | modulator | Details |
Desflurane | approved | yes | target | positive allosteric modulator | Details |
Alprazolam | approved, illicit, investigational | yes | target | positive allosteric modulator | Details |
Butabarbital | approved, illicit | yes | target | positive allosteric modulator | Details |
Chlordiazepoxide | approved, illicit, investigational | yes | target | positive allosteric modulator | Details |
Clobazam | approved, illicit | yes | target | positive allosteric modulator | Details |
Clonazepam | approved, illicit | yes | target | positive allosteric modulator | Details |
Clorazepic acid | approved, illicit | yes | target | positive allosteric modulator | Details |
Lorazepam | approved | yes | target | positive allosteric modulator | Details |
Ethchlorvynol | approved, illicit, withdrawn | yes | target | positive allosteric modulator | Details |
Enflurane | approved, investigational, vet_approved | yes | target | potentiator | Details |
Temazepam | approved, investigational | yes | target | positive allosteric modulator | Details |
Butalbital | approved, illicit | yes | target | positive allosteric modulator | Details |
Etomidate | approved | yes | target | positive allosteric modulator | Details |
Talbutal | approved, illicit | yes | target | positive allosteric modulator | Details |
Pentobarbital | approved, investigational, vet_approved | yes | target | positive allosteric modulator | Details |
Meprobamate | approved, illicit | yes | target | positive allosteric modulator | Details |
Eszopiclone | approved, investigational | yes | target | positive allosteric modulator | Details |
Metharbital | withdrawn | yes | target | positive allosteric modulator | Details |
Isoflurane | approved, vet_approved | yes | target | positive allosteric modulator | Details |
Primidone | approved, vet_approved | yes | target | positive allosteric modulator | Details |
Halazepam | approved, illicit, withdrawn | yes | target | positive allosteric modulator | Details |
Propofol | approved, investigational, vet_approved | yes | target | positive allosteric modulator | Details |
Diazepam | approved, illicit, investigational, vet_approved | yes | target | positive allosteric modulator | Details |
Oxazepam | approved | yes | target | positive allosteric modulator | Details |
Methoxyflurane | approved, investigational, vet_approved, withdrawn | yes | target | positive allosteric modulator | Details |
Methyprylon | approved, illicit, withdrawn | yes | target | positive allosteric modulator | Details |
Halothane | approved, vet_approved | yes | target | positive allosteric modulator | Details |
Flumazenil | approved | yes | target | positive allosteric modulator | Details |
Estazolam | approved, illicit | yes | target | positive allosteric modulator | Details |
Sevoflurane | approved, vet_approved | yes | target | agonist | Details |
Glutethimide | approved, illicit | yes | target | positive allosteric modulator | Details |
Prazepam | approved, illicit | yes | target | positive allosteric modulator | Details |
Quazepam | approved, illicit | yes | target | positive allosteric modulator | Details |
Amoxapine | approved | unknown | target | binder | Details |
Prasterone | approved, investigational, nutraceutical | unknown | target | antagonist | Details |
Thiocolchicoside | experimental | yes | target | antagonist | Details |
Stiripentol | approved | yes | target | agonistpositive allosteric modulator | Details |
Taurine | approved, nutraceutical | yes | target | agonist | Details |
Lamotrigine | approved, investigational | unknown | target | antagonistinducer | Details |
Apalutamide | approved, investigational | no | target | antagonist | Details |
Brexanolone | approved, investigational | yes | target | positive allosteric modulator | Details |
Memantine | approved, investigational | unknown | target | binder | Details |
Medroxyprogesterone acetate | approved, investigational | unknown | target | inhibitor | Details |
Phenytoin | approved, vet_approved | unknown | target | | Details |
Midazolam | approved, illicit | yes | target | positive allosteric modulator | Details |
Flurazepam | approved, illicit, investigational | yes | target | positive allosteric modulator | Details |
Triazolam | approved, investigational | yes | target | positive allosteric modulator | Details |
Bromazepam | approved, illicit, investigational | yes | target | positive allosteric modulator | Details |
Nitrazepam | approved | yes | target | positive allosteric modulator | Details |
Camazepam | experimental, illicit | yes | target | positive allosteric modulator | Details |
Delorazepam | experimental, illicit | yes | target | positive allosteric modulator | Details |
Flunitrazepam | approved, illicit | yes | target | positive allosteric modulator | Details |
Etizolam | experimental | yes | target | positive allosteric modulator | Details |
Medazepam | experimental | yes | target | positive allosteric modulator | Details |
Doxefazepam | experimental | yes | target | positive allosteric modulator | Details |
Lormetazepam | approved | yes | target | positive allosteric modulator | Details |
Nordazepam | experimental | yes | target | positive allosteric modulator | Details |
Adinazolam | experimental | yes | target | positive allosteric modulator | Details |
Ethyl loflazepate | experimental, illicit | yes | target | positive allosteric modulator | Details |
Cloxazolam | experimental | yes | target | positive allosteric modulator | Details |
Clotiazepam | approved, illicit | yes | target | positive allosteric modulator | Details |
Ketazolam | approved | yes | target | positive allosteric modulator | Details |
Cinolazepam | experimental | yes | target | positive allosteric modulator | Details |
Brotizolam | investigational, withdrawn | yes | target | positive allosteric modulator | Details |
Pinazepam | experimental | yes | target | positive allosteric modulator | Details |
Loprazolam | experimental | yes | target | positive allosteric modulator | Details |
Oxazepam acetate | experimental | yes | target | positive allosteric modulator | Details |
1,2-Benzodiazepine | approved, investigational | unknown | target | positive allosteric modulator | Details |
Cinazepam | experimental | yes | target | positive allosteric modulator | Details |
Bentazepam | experimental | yes | target | positive allosteric modulator | Details |
Mexazolam | experimental | yes | target | positive allosteric modulator | Details |
Remimazolam | approved, investigational | yes | target | positive allosteric modulator | Details |
Ganaxolone | approved, investigational | yes | target | positive allosteric modulator | Details |
Zuranolone | approved, experimental | yes | target | positive allosteric modulator | Details |
Adipiplon | investigational | yes | target | partial agonist | Details |
5,7,2′-trihydroxy-6,8-dimethoxyflavone | experimental | unknown | target | ligand | Details |
Lamotrigine | approved, investigational | unknown | target | inhibitor | Details |
Olanzapine | approved, investigational | no | target | inhibitor | Details |
Mexazolam | experimental | yes | target | ligand | Details |
Oxazepam | approved | yes | target | ligand | Details |
Alprazolam | approved, illicit, investigational | yes | target | ligand | Details |
Lorazepam | approved | yes | target | ligand | Details |
Temazepam | approved, investigational | unknown | target | ligand | Details |
Chlordiazepoxide | approved, illicit, investigational | yes | target | ligand | Details |
Clorazepic acid | approved, illicit | yes | target | ligand | Details |
Midazolam | approved, illicit | yes | target | ligand | Details |
Flurazepam | approved, illicit, investigational | yes | target | ligand | Details |
Diazepam | approved, illicit, investigational, vet_approved | yes | target | ligand | Details |
Triazolam | approved, investigational | yes | target | ligand | Details |
Clonazepam | approved, illicit | yes | target | ligand | Details |
Estazolam | approved, illicit | yes | target | ligand | Details |
Bromazepam | approved, illicit, investigational | yes | target | ligand | Details |
Nitrazepam | approved | yes | target | ligand | Details |
Clobazam | approved, illicit | yes | target | ligand | Details |
Camazepam | experimental, illicit | yes | target | ligand | Details |
Delorazepam | experimental, illicit | yes | target | ligand | Details |
Flunitrazepam | approved, illicit | yes | target | ligand | Details |
Prazepam | approved, illicit | yes | target | ligand | Details |
Etizolam | experimental | yes | target | ligand | Details |
Medazepam | experimental | yes | target | ligand | Details |
Doxefazepam | experimental | yes | target | ligand | Details |
Lormetazepam | approved | yes | target | ligand | Details |
Nordazepam | experimental | yes | target | ligand | Details |
Adinazolam | experimental | yes | target | ligand | Details |
Halazepam | approved, illicit, withdrawn | unknown | target | ligand | Details |
Ethyl loflazepate | experimental, illicit | yes | target | ligand | Details |
Cloxazolam | experimental | yes | target | ligand | Details |
Clotiazepam | approved, illicit | yes | target | ligand | Details |
Ketazolam | approved | yes | target | ligand | Details |
Cinolazepam | experimental | yes | target | ligand | Details |
Brotizolam | investigational, withdrawn | yes | target | ligand | Details |
Pinazepam | experimental | yes | target | ligand | Details |
Loprazolam | experimental | unknown | target | ligand | Details |
Quazepam | approved, illicit | yes | target | ligand | Details |
Oxazepam acetate | experimental | yes | target | ligand | Details |
1,2-Benzodiazepine | approved, investigational | unknown | target | ligand | Details |
Cinazepam | experimental | yes | target | ligand | Details |
Bentazepam | experimental | yes | target | ligand | Details |
Remimazolam | approved, investigational | yes | target | ligand | Details |
Zonisamide | approved, investigational | unknown | target | binder | Details |