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Deleobuvir
go.drugbank.com/drugs/DB14850InvestigationalDeleobuvir is under investigation in clinical trial NCT01983566 (Effect of Food and Increased Gastric pH Value on Bioavailability of a Single Dose of BI 207127 in Healthy Caucasian and Japanese Subjects
Categories: Heterocyclic Compounds, 2-RingGO-203-2C
go.drugbank.com/drugs/DB15008InvestigationalGO-203-2C is under investigation in clinical trial NCT02204085 (A Phase I/II Trial of the MUC1 Inhibitor, GO-203-2C in Patients With Relapsed or Refractory Acute Myeloid Leukemia).
Synonyms: Acetyl-D-arginyl-D-arginyl-D-arginyl-D-arginyl-D-arginyl-D-arginyl-D-arginyl-D-arginyl-D-arginyl-D-cysteinyl-D-glutaminyl-D-cysteinyl-D-arginyl-D-arginyl-D-lysyl-dasparaginylamide disulfideIlacirnon
go.drugbank.com/drugs/DB16066InvestigationalIlacirnon (CCX-140) is under investigation in clinical trial NCT01440257 (A Study to Evaluate the Effect of CCX140-B on Urinary Albumin Excretion in Subjects With Type 2 Diabetes and Albuminuria).
Synonyms: 4-Chloro-N-[5-methyl-2-(7H-pyrrolo[2,3-d]pyrimidin-4-ylcarbonyl)-3-pyridinyl]-3-(trifluoromethyl)benzenesulfonamideIndoramin
go.drugbank.com/drugs/DB08950ApprovedWithdrawnIt is a selective alpha-1 adrenergic antagonist with no reflex tachycardia and direct myocardial depression action. … Indoramin is a discontinued piperidine antiadrenergic drug with the trade names Baratol and Doralese.
Categories: Peripheral alpha-1 blockers, Heterocyclic Compounds, 1-RingMivebresib
go.drugbank.com/drugs/DB21300InvestigationalMivebresib is a small molecule drug. … The usage of the INN stem '-bresib' in the name indicates that Mivebresib is a inhibitor of the bromodomain and extra-terminal motif (BET) family of bromodomain (BRD) protein, antineoplastic.
Categories: Heterocyclic Compounds, 1-RingPhenamazoline
go.drugbank.com/drugs/DB19509ExperimentalPhenamazoline is a small molecule drug. The usage of the INN stem '-azoline' in the name indicates that Phenamazoline is a antihistaminic or local vasoconstrictor, antazoline derivative. … Phenamazoline has a monoisotopic molecular weight of 175.11 Da.
Glaspimod
go.drugbank.com/drugs/DB19609ExperimentalGlaspimod is a small molecule drug. The usage of the INN stem '-imod' in the name indicates that Glaspimod is a immunomodulator, both stimulant/suppressive and stimulant. … Glaspimod has a monoisotopic molecular weight of 1170.5 Da.
Mifentidine
go.drugbank.com/drugs/DB19721ExperimentalMifentidine is a small molecule drug. The usage of the INN stem '-tidine' in the name indicates that Mifentidine is a histamine- H2-receptor antagonist, cimetidine derivative. … Mifentidine has a monoisotopic molecular weight of 228.14 Da.
Categories: Cytochrome P-450 CYP1A2 Inhibitors, Heterocyclic Compounds, 1-RingRazaxaban
go.drugbank.com/drugs/DB19834ExperimentalRazaxaban is a small molecule drug. The usage of the INN stem '-xaban' in the name indicates that Razaxaban is a blood coagulation factor XA inhibitor, antithrombotic. … Razaxaban has a monoisotopic molecular weight of 528.16 Da.
Categories: Heterocyclic Compounds, 1-RingIvarimod
go.drugbank.com/drugs/DB19605ExperimentalIvarimod is a small molecule drug. The usage of the INN stem '-imod' in the name indicates that Ivarimod is a immunomodulator, both stimulant/suppressive and stimulant. … Ivarimod has a monoisotopic molecular weight of 512.33 Da.