| DB00486 | Nabilone | approved, investigational | yes | partial agonist | Details |
| DB00470 | Dronabinol | approved, illicit | yes | agonist | Details |
| DB06202 | Lasofoxifene | approved, investigational | unknown | inverse agonist | Details |
| DB02955 | Ricinoleic acid | experimental | unknown | | Details |
| DB09061 | Cannabidiol | approved, investigational | unknown | antagonist | Details |
| DB14011 | Nabiximols | investigational | yes | | Details |
| DB14009 | Medical Cannabis | experimental, investigational | unknown | | Details |
| DB11755 | Tetrahydrocannabivarin | investigational | unknown | partial agonist | Details |
| DB16321 | S-777469 | investigational | unknown | agonist | Details |