| DB02122 | 4-iodo-acetamido phenylboronic acid | experimental | unknown | | Details |
| DB02816 | 7-(1-Methyl-1,2,3-Triazol-4-Yl)-6-Formyl-2,7-Dihydro-[1,4]Thiazepine-3-Carboxylic Acid, Brl42715, C6-(N1-Methyl-1,2,3-Triazolylmethylene)Penem | experimental | unknown | | Details |
| DB02876 | 3-(4-carbamoyl-1-carboxy-2-methylsulfonyl-buta-1,3-dienylamino)-indolizine-2-carboxylic acid | experimental | unknown | | Details |
| DB03970 | (7R)-7-(6,7-Dihydro-5H-cyclopenta[d]imidazo[2,1-b][1,3]thiazol-2-yl)-2,7-dihydro-1,4-thiazepine-3,6-dicarboxylic acid | experimental | unknown | | Details |
| DB04123 | (P-Iodophenylacetylamino)Methylphosphinic Acid | experimental | unknown | | Details |
| DB08109 | (1S,4R,7AR)-4-BUTOXY-1-[(1R)-1-FORMYLPROPYL]-2,4,5,6,7,7A-HEXAHYDRO-1H-ISOINDOLE-3-CARBOXYLIC ACID | experimental | unknown | | Details |
| DB08110 | (1R,4S,7AS)-1-(1-FORMYLPROP-1-EN-1-YL)-4-METHOXY-2,4,5,6,7,7A-HEXAHYDRO-1H-ISOINDOLE-3-CARBOXYLIC ACID | experimental | unknown | | Details |
| DB09060 | Avibactam | approved | yes | inhibitor | Details |
| DB12107 | Vaborbactam | approved, investigational | yes | inhibitor | Details |
| DB12377 | Relebactam | approved, investigational | yes | inhibitor | Details |