Gephyrin

BE0002652ProteinHumansGPHN

Microtubule-associated protein involved in membrane protein-cytoskeleton interactions. It is acted on by 3 drugs in DrugBank.

Gene name
GPHN
UniProtKB entry
Q9NQX3Swiss-Prot
Cellular location
Postsynaptic cell membrane
Residues / weight
736 residues · 79,748 Da
Also known as
GPH · KIAA1385

Resolves to

Protein
UniProtQ9NQX3UniProt nameGEPH_HUMAN
Gene
HGNCHGNC:15465NCBI Gene10243GeneCardsGPHN
Pharmacology
KEGGhsa:10243
Structure
PDB1JLJ
Drugs

What you can answer from here — as of September 07, 2019

3DrugsApproved to experimental, with action, bond type and pharmacological action
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12GO termsFunction, process and component, as structured annotations
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3Pfam domainsDomain architecture mapped to Pfam families and clans
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17+ReferencesStructured and connected to the statements they support
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Which approved drugs act on Gephyrin, how selective are they, and which programs against it are still in active trials?

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