G protein-coupled receptor kinase 5
BE0013072ProteinHumansGRK5
Serine/threonine kinase that phosphorylates preferentially the activated forms of a variety of G protein-coupled receptors (GPCRs). It is acted on by 1 drug in DrugBank.
- Gene name
- GRK5
- UniProtKB entry
- P34947Swiss-Prot
- Cellular location
- Cytoplasm
- Residues / weight
- 590 residues · 67,786 Da
- Also known as
- 2.7.11.16 · G protein-coupled receptor kinase GRK5 · GPRK5
Resolves to
Pharmacology
Drugs
What you can answer from here — as of September 03, 2024
Which approved drugs act on G protein-coupled receptor kinase 5, how selective are they, and which programs against it are still in active trials?
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