Adrenergic beta-3 Receptor Agonists

Name
Adrenergic beta-3 Receptor Agonists
Accession Number
DBCAT001740  (DBCAT003499)
Description

Compounds that bind to and activate ADRENERGIC BETA-3 RECEPTORS.

Drugs
DrugDrug Description
AmibegronInvestigated for use/treatment in depression, irritable bowel syndrome (IBS), and obesity.
ArbutamineUsed to elicit acute cardiovascular responses (cardiac stumulant), similar to those produced by exercise, in order to aid in diagnosing the presence or absence of coronary artery disease (CAD) in...
CeliprololA beta-blocker for the management of hypertension and angina pectoris.
DipivefrinA prodrug of epinephrine used in ophthalmic solutions to reduce intraocular pressure in chronic open-angle glaucoma.
DroxidopaA medication used to treat symptomatic neurogenic orthostatic hypotension (nOH) caused by dopamine beta-hydroxylase deficiency, non-diabetic autonomic neuropathy and primary autonomic failure caused by conditions such as Parkinson's disease.
EpinephrineA hormone and neurotransmitter used to treat allergic reactions, to restore cardiac rhythm, and to control mucosal congestion, glaucoma, and asthma.
MirabegronA beta-3 adrenergic agonist used to treat overactive bladder and neurogenic detrusor overactivity.
NorepinephrineA sympathomimetic used in the control of blood pressure during various hypotensive states and as an adjunct treatment during cardiac arrest.
RacepinephrineA bronchodilator used to treat intermittent asthma.
RitobegronRitobegron is under investigation in clinical trial NCT02256735 (Study to Investigate the Effect of KUC 7483 CL on the QT/QTc Interval of the ECG in Comparison to Placebo and Moxifloxacin...
SolabegronInvestigated for use/treatment in diabetes mellitus type 2, irritable bowel syndrome (IBS), and urinary incontinence.
VibegronA beta-3 adrenergic agonist the treatment of overactive bladder (OAB) with symptoms of urge urinary incontinence, urgency, and urinary frequency in adults.
Drugs & Drug Targets
DrugTargetType
AmibegronBeta-3 adrenergic receptortarget
ArbutamineBeta-1 adrenergic receptortarget
ArbutamineBeta-2 adrenergic receptortarget
ArbutamineBeta-3 adrenergic receptortarget
CeliprololBeta-2 adrenergic receptortarget
CeliprololBeta-1 adrenergic receptortarget
CeliprololBeta-3 adrenergic receptortarget
CeliprololAlpha-2A adrenergic receptortarget
CeliprololAlpha-2B adrenergic receptortarget
CeliprololAlpha-2C adrenergic receptortarget
CeliprololCytochrome P450 2D6enzyme
CeliprololAlpha-2 adrenergic receptorstarget
DipivefrinAlpha-2A adrenergic receptortarget
DipivefrinCholinesterasetarget
DipivefrinBeta-2 adrenergic receptortarget
DipivefrinAlpha-1A adrenergic receptortarget
DipivefrinAcetylcholinesterasetarget
DipivefrinBeta-1 adrenergic receptortarget
DroxidopaSodium-dependent noradrenaline transportertransporter
DroxidopaMonocarboxylate transporter 10transporter
DroxidopaAromatic-L-amino-acid decarboxylaseenzyme
DroxidopaBeta-3 adrenergic receptortarget
DroxidopaBeta-2 adrenergic receptortarget
DroxidopaBeta-1 adrenergic receptortarget
DroxidopaAlpha-2C adrenergic receptortarget
DroxidopaAlpha-2B adrenergic receptortarget
DroxidopaAlpha-2A adrenergic receptortarget
DroxidopaAlpha-1D adrenergic receptortarget
DroxidopaPhenylalanine-4-hydroxylasetarget
DroxidopaAlpha-1A adrenergic receptortarget
DroxidopaAlpha-1B adrenergic receptortarget
EpinephrineCytochrome P450 2C9enzyme
EpinephrineSolute carrier family 22 member 1transporter
EpinephrineAlpha-1B adrenergic receptortarget
EpinephrineAlpha-1D adrenergic receptortarget
EpinephrineAlpha-2A adrenergic receptortarget
EpinephrineAlpha-2B adrenergic receptortarget
EpinephrineTumor necrosis factortarget
EpinephrineCatechol O-methyltransferaseenzyme
EpinephrineMonoamine oxidaseenzyme
EpinephrineSolute carrier family 22 member 2transporter
EpinephrineBeta-2 adrenergic receptortarget
EpinephrineBeta-1 adrenergic receptortarget
EpinephrineAlpha-1A adrenergic receptortarget
EpinephrineCytochrome P450 3A4enzyme
MirabegronSolute carrier organic anion transporter family member 1A2transporter
MirabegronATP-dependent translocase ABCB1transporter
MirabegronCytochrome P450 2D6enzyme
MirabegronCytochrome P450 3A4enzyme
MirabegronBeta-1 adrenergic receptortarget
MirabegronSolute carrier family 22 member 3transporter
MirabegronSolute carrier family 22 member 2transporter
MirabegronSolute carrier family 22 member 1transporter
MirabegronUDP-glucuronosyltransferase 1A8enzyme
MirabegronUDP-glucuronosyltransferase 1A3enzyme
MirabegronUDP-glucuronosyltransferase 2B7enzyme
MirabegronBeta-3 adrenergic receptortarget
MirabegronCholinesteraseenzyme
MirabegronAlpha-1-acid glycoprotein 1carrier
MirabegronAlbumincarrier
NorepinephrineChromaffin granule amine transportertarget
NorepinephrineSynaptic vesicular amine transportertarget
NorepinephrineSodium-dependent noradrenaline transportertransporter
NorepinephrinePOU domain, class 5, transcription factor 1transporter
NorepinephrineSolute carrier family 22 member 1transporter
NorepinephrineOrganic cation/carnitine transporter 2transporter
NorepinephrineSolute carrier family 22 member 3transporter
NorepinephrineSolute carrier family 22 member 2transporter
NorepinephrineBeta-3 adrenergic receptortarget
NorepinephrineBeta-2 adrenergic receptortarget
NorepinephrineBeta-1 adrenergic receptortarget
NorepinephrineAlpha-2C adrenergic receptortarget
NorepinephrineAlpha-2B adrenergic receptortarget
NorepinephrineAlpha-2A adrenergic receptortarget
NorepinephrineAlpha-1D adrenergic receptortarget
NorepinephrineAlpha-1B adrenergic receptortarget
NorepinephrineAlpha-1A adrenergic receptortarget
NorepinephrinePhenylalanine-4-hydroxylasetarget
RacepinephrineBeta-3 adrenergic receptortarget
RacepinephrineAlpha-1D adrenergic receptortarget
RacepinephrineBeta-2 adrenergic receptortarget
RacepinephrineBeta-1 adrenergic receptortarget
RacepinephrineAlpha-2C adrenergic receptortarget
RacepinephrineAlpha-2B adrenergic receptortarget
RacepinephrineAlpha-2A adrenergic receptortarget
RacepinephrineAlpha-1B adrenergic receptortarget
RacepinephrineAlpha-1A adrenergic receptortarget
RitobegronBeta-3 adrenergic receptortarget
SolabegronBeta-3 adrenergic receptortarget
VibegronBeta-3 adrenergic receptortarget
VibegronCytochrome P450 3A4enzyme
VibegronATP-dependent translocase ABCB1transporter